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[(1-methyl-1H-imidazol-2-yl)methyl](2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amine
N,N-dimethyl-5-(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidin-2-yl)thiophene-2-carboxamide
ethyl 1-(3,4-dimethoxybenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
1-{2-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-methoxy-2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-4-cyclopentylpiperazin-2-one
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
2-(methylsulfanyl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-(4-chloro-2-methylphenoxy)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
3-(3-methoxybenzoyl)-9-(1-methylpiperidin-4-yl)-3,9-diazaspiro[5.5]undecane
3-benzoyl-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine
1-(4-methoxyphenyl)-4-[1-(4-methylpent-3-en-1-yl)piperidin-3-yl]piperazine
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)pyrazine-2-carboxamide
N-(2-methoxyethyl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(propan-2-yl)propanamide
3-{3-methyl-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-{1-[(4-fluorophenyl)methyl]-5-(2-methoxypyridin-3-yl)-1H-1,2,4-triazol-3-yl}acetamide
4-(cyclopropylamino)-N-(cyclopropylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-methoxy-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-1-methyl-1H-pyrazole-4-carboxamide
N2-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-N1-ethylpyrrolidine-1,2-dicarboxamide
(1R,5R)-6-methyl-3-[(3-methylthiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-chlorophenyl)-4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]piperazine
2-acetamido-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
3-{2-[1-(1-benzofuran-5-carbonyl)piperidin-2-yl]ethyl}phenol
3-ethyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-2-(methylamino)acetamide
1-methyl-5-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazole
1-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-1,7-dimethyl-2,4-dioxo-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-5-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
5-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-(5-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}furan-2-yl)benzonitrile
9-(1H-indol-5-ylmethyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,2,2,6,6-pentamethylpiperidin-4-amine
4-[(benzyloxy)methyl]-3-methyl-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(2-methoxyphenyl)-2-(4-methyl-1,2,3-thiadiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
3-(piperidin-4-ylmethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}benzamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
4-(2,5-dimethoxyphenyl)-2-[5-methyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N-[(6-hydroxypyrimidin-4-yl)methyl]-2,5,7-trimethylquinoline-4-carboxamide
4-(4-chloro-2-fluorobenzoyl)-1-(1H-indazol-5-yl)piperazin-2-one
1-(2-cyclohexylethyl)-3-hydroxy-3-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-ylmethyl)piperidin-2-one
2-{4-[(3-methylthiophen-2-yl)methyl]morpholin-3-yl}acetic acid
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-[1-(pyrimidin-4-yl)ethyl]acetamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one