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3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-methoxypyridin-3-yl)-3-methylurea
8-fluoro-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]quinoline
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
4-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-1-(propan-2-yl)pyrrolidin-2-one
(1S,5R)-N-(3,4-difluorophenyl)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-amino-7-methoxy-4-(oxolan-3-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
3-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-6-methyl-1,4-dihydroquinolin-4-one
N-[2-(2,4-dimethylphenoxy)ethyl]-4-(2-methoxyacetamido)-N-methylbenzamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
2-{3-[2-amino-3-cyano-6-(trimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenoxy}acetamide
2-fluoro-6-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)phenol
3-butyl-4-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-1-methylpiperazin-2-one
4-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
3-(2-hydroxy-3-methoxybenzamido)-4-(3-methylpiperidin-1-yl)benzamide
3-(4-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}piperazin-1-yl)propanamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(2-methoxyphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
6-ethyl-N,1,5-trimethyl-2-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2-(pyridin-2-yl)pyrimidine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
({4-ethyl-5-[1-(isoquinoline-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,2-dimethyl-3-[(pyridin-2-ylmethyl)amino]benzamide
N,N-dimethyl-2-{[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]amino}ethane-1-sulfonamide
2-(4-fluorophenyl)-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-6-carboxamide
ethyl 4-{[(7-fluoro-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino}piperidine-1-carboxylate
1-[(4-chlorophenyl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(2,4-dimethylphenyl)-4-(hydroxymethyl)-4-(2-phenylethyl)piperidine-1-carboxamide
1-cyclopentyl-4-{[2-(1-methylpiperidin-4-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-oxo-N-phenylacetamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methanesulfonylpiperidin-4-amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
3-chloro-2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-1H-indole
4-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-amine
2-{3-methyl-5-[5-(oxolan-2-yl)thiophen-2-yl]-1H-1,2,4-triazol-1-yl}pyridine
2-(2-{[3-(dimethyl-1,2-oxazol-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(4aR,7aS)-N,N-dimethyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[2-(morpholin-4-yl)ethyl]-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
{4-[(4-methoxyphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidin-4-yl}methanol
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-(1,3-thiazol-2-ylmethyl)piperidin-3-ol
1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}piperidine-2-carboxylic acid
(4aS,7aR)-1-[2-(2-chlorophenoxy)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
2-(4-acetyl-1,4-diazepan-1-yl)-2-[5-chloro-2-(propan-2-yloxy)phenyl]acetic acid