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N-{[8-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}cyclopropanamine
methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})(quinoxalin-2-ylmethyl)amine
3-[2-(1H-indol-5-yl)ethyl]-1λ6-thiolane-1,1-dione
2-[3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)phenoxy]acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]urea
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
9-(2-chloro-5-fluorobenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1-(4-ethoxy-2-fluorophenyl)-3-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-amine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
3-{2-[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}propanamide
N-cyclohexyl-3-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
3-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3,4-dihydropteridin-4-one
2-(4-fluorophenyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-phenyl-5-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
N-[1-(thian-4-yl)piperidin-4-yl]-1,3-benzothiazole-6-carboxamide
N-cyclopentyl-5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-ethyl-2-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]quinoline-4-carboxamide
(1R,5R)-N-(furan-2-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(1H-pyrazol-3-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
N-[2-(dimethylamino)ethyl]-N-ethyl-1-[2-(naphthalen-1-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)propanamide
N-butyl-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydroquinoline-2-carboxamide
3-{[(4aS,7aR)-4-(carboxymethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]amino}propanoic acid
3-(methanesulfonylmethyl)-1-{[2-(methylsulfanyl)phenyl]methyl}piperidine
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
8-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-oxazole-5-carboxamide
4-[(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)methyl]-N-(1,2,3-thiadiazol-5-yl)benzamide
5-(2-methylpropyl)-1'-(quinoxalin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2-fluorophenyl)methyl]-3-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}propanamide
1-(2,4-dimethoxyphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{4-[4-(azocane-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(oxan-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
1-(oxolane-3-carbonyl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[4-(4-fluorophenyl)butanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-(4-{[(1R,2S)-2-phenylcyclopropyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
2-(3-chlorophenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
1-(4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-methoxy-2-(3-{1-[(3-methylpyridin-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
4-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]oxane-4-carbonitrile
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-fluoro-4-methylphenyl)methyl]piperidine
N-[(4-hydroxyphenyl)methyl]-1-(methoxymethyl)-N-(pyridin-4-ylmethyl)cyclobutane-1-carboxamide