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3-(3-methyl-1H-pyrazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
7-methanesulfonyl-4-methyl-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)azepan-1-yl]quinazoline
3-(3-hydroxy-3-methylbutyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(2-methoxy-5-methylbenzenesulfonamido)acetic acid
2-(1,6-dimethyl-1H-indole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-propylpiperazine
4-ethyl-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-phenylbenzoyl)-1-(propane-1-sulfonyl)piperidine
(2R)-N-(6-chloro-2-methylpyridin-3-yl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
methyl 3-(oxolane-2-amido)-5-[(pentan-3-yl)amino]-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(3-fluorophenyl)-2-oxo-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N,1-dimethyl-2-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}imidazolidine-4-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
2-(pyridin-3-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-4-(2-propylpyrrolidine-1-carbonyl)-1,3-oxazole
1-[2-(piperidin-1-yl)acetyl]-4-(pyrimidin-2-yl)-1,4-diazepane-6-carboxylic acid
4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
2-(4-fluoro-3-methylphenyl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]quinoxaline-2-carboxamide
(1R,9aR)-1-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxymethyl]-octahydro-1H-quinolizine
N-({1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
N-[3-(3-fluorophenyl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
2-(propylsulfanyl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
1-(4-fluorophenyl)-4-{5-[(methylsulfanyl)methyl]pyridin-2-yl}-1,4-diazepane
(3S,4S)-4-[({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]piperidin-3-ol
N-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-[4-(3-methoxyphenyl)phenyl]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-[({[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)methyl]-6-methyl-3,4-dihydropyrimidin-4-one
2-(4-fluorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
5-methoxy-2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridin-4-ol
1-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
2-{1-[(4-methylphenyl)methyl]-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
3-{5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-3-yl}pyridine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pent-4-enamide
3-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamido]-3-(furan-2-yl)propanoic acid
2-{4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]piperidine-1-carbonyl}pyridine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(piperidin-4-yl)benzamide
1-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidine-1-carbonyl]cyclopropane-1-carbonitrile
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
N-[(3R,4S)-4-(propan-2-yl)-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
N-[3-(cyclohexyloxy)propyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
2-(3-phenylpropyl)-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-ol
N,N-bis(2-ethoxyethyl)-2-methylthieno[2,3-d]pyrimidin-4-amine
N-({3-methyl-7-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxolane-2-carboxamide