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8-(2-amino-6-methoxypyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclopropane-1-carboxamide
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][(3-{[1-(quinoline-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-3-phenylpiperazine
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
3-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(4-methanesulfonylphenyl)urea
3-methyl-6-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridazine
N-benzyl-N-methyl-2-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2,3-dihydro-1H-inden-2-amine
(2S,4R)-N-(diphenylmethyl)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{3-[(pyridin-3-yl)amino]propyl}butanamide
N-{5-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]-2-methylphenyl}cyclopropanecarboxamide
(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanamine
2,2-dimethyl-6-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]-3,4-dihydro-2H-pyran-4-one
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-(2-methylphenyl)pyrrolidin-3-ol
1-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-ethyl-1H-pyrazole-4-carboxamide
(1S,5R)-3-(2-phenylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2-chloro-3,4-dimethoxyphenyl)methyl](methyl)(quinoxalin-2-ylmethyl)amine
1-tert-butyl-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
[(3R,4R)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(1S,5R)-3-(isoquinolin-1-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(3,5-difluoropyridine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-dimethoxyphenyl)-1-(4-phenylbenzoyl)piperidin-3-amine
2-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]furan-3-carboxamide
10-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
2-(2-{1-[2-(3,4-dimethylphenoxy)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-(2-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]propanoic acid
1-ethyl-N-methyl-3-(2-methylpropyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
6-(2-cyclopropyl-1,3-benzoxazol-5-yl)hexan-1-ol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
4-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-diazepane-1-carbaldehyde
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
N,3,6-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrazin-2-amine
1-(3-methyl-1H-pyrazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-(2,5-dimethylphenyl)-3-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]propanamide
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-oxo-6-(3,4,5-trimethoxyphenyl)-1,4-dihydroquinoline-3-carboxylic acid
N3-benzyl-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,3-diphenylpiperidine
methyl 4-{4-[3-(ethylcarbamoyl)pyridin-2-yl]piperazin-1-yl}benzoate
[(3-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)sulfamoyl]dimethylamine
4-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-7-fluoroquinazoline
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
6-(2-aminoethyl)-2-(4-{[3-(trifluoromethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one