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N-[1-(3-methylpyridin-2-yl)propan-2-yl]thian-4-amine
1-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-indole-6-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrrole-3-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-N-phenylpyrimidin-2-amine
(1S,6R)-3-methyl-9-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
1-(2-{4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1-benzofuran-2-sulfonamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[2-(furan-2-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
4-({[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)carbamoyl}amino)-N-(2-methoxyethyl)benzamide
7-methyl-2-(2,3,4-trifluorobenzenesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[5-chloro-2-(propan-2-yloxy)phenyl]-6-methylpyridazine
4-(4-ethyl-1H-pyrazol-5-yl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-1,4-diazepane
ethyl 4-(2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
2-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)-1H-indole
1-[(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-{[(2S,4S)-4-fluoro-1-[2-(2-methylphenyl)acetyl]pyrrolidin-2-yl]methyl}morpholine-4-carboxamide
5-{[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
3-hexyl-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-(3-methylthiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,3-dimethyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1'-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)spiro[indene-1,4'-piperidine]
N-methyl-5-phenoxy-N-(1H-pyrazol-3-ylmethyl)furan-2-carboxamide
3-[({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}oxy)methyl]pyridine
4-(4-methyl-1H-pyrazol-1-yl)-1-[(2E)-3-phenylprop-2-enoyl]piperidine-4-carboxylic acid
3-methoxy-2-[4-(1-methoxyethyl)phenyl]pyridin-4-amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]furan-2-carboxamide
2-[5-({2,5-dimethyl-3-[(3-methylpiperidin-1-yl)methyl]phenyl}methyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
methyl 4-({2-oxo-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]azepan-1-yl}methyl)benzoate
{2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazol-4-yl}methanol
2-ethoxy-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)acetamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-ethylpiperidine-3-carboxylic acid
[(dimethyl-1,2-oxazol-4-yl)methyl][4-(1H-indol-3-yl)butan-2-yl]amine
2-(2,5-difluorophenyl)-N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-({5-[(3-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
(butan-2-yl)[(4-methylphenyl)methyl](1,3-thiazol-2-ylmethyl)amine
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[3-(methylsulfanyl)propyl]carbamoyl}pyrrolidine-2-carboxylate
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-{1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl}acetamide
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
N,N,8-trimethyl-2-[2-(3-methylbutyl)pyrimidin-5-yl]quinoline-4-carboxamide
2-(3-methoxypropyl)-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
5-[1-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]benzonitrile
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide