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5-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}-3-methylpyridin-2-amine
4-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]morpholine
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(4-chlorophenyl)methyl]piperidine
5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-phenylpropyl)piperidin-4-yl]oxy}benzamide
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}azepan-2-one
N-(furan-2-ylmethyl)-5-{[(1-hydroxycyclohexyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)(quinolin-4-ylmethyl)amine
N-[2-(2-methoxyphenyl)ethyl]-2-[(prop-2-yn-1-yl)amino]acetamide
(3aR,7aS)-5-methyl-2-[1-(pyridine-2-carbonyl)piperidine-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-methyl-8-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-2,8-diazaspiro[4.5]decane
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][(4-fluorophenyl)methyl]amino}butan-1-ol
2-tert-butyl-6-(2,4,5-trimethoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(3aS,6aR)-5-[(3-fluorophenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(2-aminoethyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)quinazolin-4-amine
5-cyclopropanecarbonyl-1'-(6-methylpyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(5-fluoro-1H-indole-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(1,3-thiazol-4-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-(cyclopropylmethyl)-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
1-methyl-2-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}-1H-indole
ethyl 5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentanoate
N-(3-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
3-{1-[1-(2-acetylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
5-tert-butyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
4-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]-2-methylphenol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2,5-dimethylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-4-yl}pyridine
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperazine
2-{2-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenoxy}ethan-1-ol
2-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)[(2,2-dimethyloxan-4-yl)methyl]methylamine
4-benzyl-6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N3-butyl-1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-(propan-2-yl)-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1H-pyrazole
N-[1-(3,4-dimethoxyphenyl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
4-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}quinazoline
4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-[2-(3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]morpholine
(2R,3R)-3-amino-1'-(2-hydroxypyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{[3-(1H-imidazol-1-yl)butanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(2-cyclohexylethyl)-3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-(2-methoxyethyl)-1-methyl-2-oxo-6-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-N-(3-hydroxypropyl)piperidine-3-carboxamide
N-(2,3-dimethylphenyl)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(3S,4S)-1-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}-4-propylpyrrolidine-3-carboxylic acid
N-(4-cyano-2,5-difluorophenyl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylpyridine-3-carboxamide