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N-(2H-1,3-benzodioxol-5-yl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-amine
N,N-diethyl-2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-sulfonamide
3-(azepane-1-sulfonyl)-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
N-(2-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)cyclopropanesulfonamide
2-{3-cyclopropyl-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazol-1-yl}pyridine
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
4-{4-[(2-aminoethoxy)methyl]phenyl}-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-({[(4-fluorophenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetamide
N-[2-(dimethylamino)ethyl]-2-hydroxy-5-methoxy-N-[(3-methylthiophen-2-yl)methyl]benzamide
N-methyl-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
6-(2,3-dimethoxyphenyl)-N4-methylpyrimidine-2,4-diamine
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanol
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propanoic acid
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-hydroxy-3-methylbutyl)-N-[1-(piperidin-1-ylmethyl)cyclopropyl]benzamide
(1S,6R)-3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 4-[({[4-(3-methoxyphenyl)-5-[(pyridin-3-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]benzoate
(4aS,7aR)-1-(5-methylpyridine-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-8-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(3,5-dimethylphenyl)piperazin-2-one
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(6-{[(2-methylphenyl)methyl]amino}pyrazin-2-yl)sulfanyl]acetic acid
{1-[(6-fluoroquinolin-2-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
3-{[({7-fluoro-2-[2-(phenylsulfanyl)ethoxy]quinolin-3-yl}methyl)amino]methyl}-1λ6-thiolane-1,1-dione
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
methyl 2-(1-{[2-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
1-(4-benzylpiperidin-1-yl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propan-1-one
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]thiophene-2-carboxamide
(2E)-N-{[1-(1-carbamoylethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-N-methyl-3-phenylprop-2-enamide
4-{1-[1-(4-methanesulfonylphenyl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
(2S,4R)-1-cyclopentyl-4-(2,5-dimethylfuran-3-amido)-N,N-diethylpyrrolidine-2-carboxamide
1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-4-hydroxypiperidine-4-carboxylic acid
3-(azepane-1-carbonyl)-1-methyl-N-(quinolin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(5-fluoro-2-methylphenyl)-2-(4-methanesulfonylphenyl)-1H-imidazole
5-(methoxymethyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)thiophene-2-carboxamide
(1R,7S)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(2-methoxyethyl)-3-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
7-(propan-2-yl)-2-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-propoxybenzamide
4-{2-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}morpholine