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1-[1-(1-cyclopropylpropan-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-[(piperidin-4-yl)amino]-N-(2,3,4-trifluorophenyl)acetamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(pyridin-3-ylmethyl)amine
5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-(propan-2-yl)-1,2,4-oxadiazole
8-(1,3-benzothiazol-2-ylmethyl)-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(5,6-dimethylpyridine-3-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-[3-(3-methylphenyl)phenyl]urea
methyl (2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
ethyl 4-[(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
8-methoxy-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
N-[7-(4-acetyl-1,4-diazepane-1-carbonyl)-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazol-5-yl]acetamide
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
4-{[(3,5-dimethoxyphenyl)methyl]amino}-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
(1S,5R)-3-benzyl-6-(dimethyl-1,3-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4-fluorophenyl)-1-(2-methylpropyl)piperidin-3-amine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-methoxyphenyl)butanamide
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
2-(4-chloro-2-methylphenoxy)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
5-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]pyridine-2-carbonitrile
1-(2-{[(3,5-difluorophenyl)methyl](methyl)amino}ethyl)piperidin-2-one
3-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)propane-1,2-diol
(2S,4R)-N-ethyl-4-[2-(pyridin-3-yl)acetamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
[(3R,4S)-1-[(4-fluoro-2-methylphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{2-methyl-4-[methyl(oxan-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
6-methoxy-1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-indole-2-carboxamide
2-(3-tert-butyl-1H-pyrazol-5-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(3S)-3-aminopyrrolidine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
(3aS,6aS)-2-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(hydroxymethyl)phenyl]-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-ethylpyrimidin-2-yl)-5-methyl-1H-indole
N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4,5-dimethyl-2-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
2-(2,3-dimethylphenoxy)-N-methyl-N-[1-(pyridin-2-yl)propyl]acetamide
(2S,4R)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-N-(thiophen-2-ylmethyl)aniline
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(trifluoromethyl)benzamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
(2S)-1-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetyl]pyrrolidine-2-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-ethylpiperazine
3-(5-chloro-2-methoxypyridin-4-yl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
3-(3-chlorophenyl)-1-(cyclopropylmethyl)-6-(oxolane-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N,N-diethyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(furan-3-ylmethyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
2-{4-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]morpholin-3-yl}acetic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(methylsulfanyl)pyrimidin-4-amine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
4-methoxy-6-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
N-(isoquinolin-5-ylmethyl)-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide