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(2S)-2-amino-N-[(1-benzylpiperidin-4-yl)methyl]-3-(4-hydroxyphenyl)-N-methylpropanamide
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-(propan-2-yl)-1,2,4-oxadiazole
2-(2-fluorophenyl)-N-[2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
6-chloro-N-cyclopentyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
methyl (2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
4-[(4-fluorophenyl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-methanesulfonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperazine-1-carboxamide
3-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-(thiophen-3-ylmethyl)benzamide
8-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-methyl-1H-imidazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
(2S,4R)-4-amino-N-[4-(pyridin-2-yl)butyl]pyrrolidine-2-carboxamide
1,9-dimethyl-4-(2-methyl-6-propylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
methyl 6-[(4-methylphenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-chloro-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
(1R,5R)-6-(3-phenoxypropyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]quinoxaline
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-phenylacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2S)-2-amino-2-[1-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]ethyl]phenol
3-(4-chlorophenyl)-4-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-[2-(3-methoxyphenyl)ethyl]-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
1-{2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]ethyl}piperidin-4-ol
(2R)-2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidine
1-tert-butyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
(1S,5R)-6-(4-chloro-3-methylbenzoyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[3-(furan-2-yl)propanoyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-(2,6-dimethoxypyridin-3-yl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
(4aR,8aR)-2-cyclobutanecarbonyl-7-[2-(3-methoxyphenoxy)ethyl]-decahydro-2,7-naphthyridin-4a-ol
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
6-(9H-fluoren-2-ylmethyl)-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
7-{imidazo[1,2-a]pyridine-3-carbonyl}-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
6-methyl-2-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-[3-(1H-imidazol-1-yl)propyl]acetamide
9-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
ethyl 4-{[(2-methanesulfonamidoethyl)carbamoyl]amino}benzoate
1-methyl-4-({5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}butanamide
9-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
5-(1-benzyl-5-methyl-1H-1,2,3-triazol-4-yl)-3-cyclopropyl-1H-1,2,4-triazole
1-(1H-imidazol-2-ylmethyl)-4-(naphthalen-2-yl)piperazine
3-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
(1R,5S,6S)-N-(furan-3-ylmethyl)-N-methyl-3-(pyridin-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-{3-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-1H-indol-1-yl}acetamide
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-propylpiperidin-3-yl}methanol
N-{[(3S,4S)-3-hydroxy-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]methyl}-2-methoxyacetamide
N-(4-methylphenyl)-3-[(1,4,6-trimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]propanamide
5-[5-(piperidine-1-carbonyl)furan-2-yl]-1,2-dihydropyridin-2-one