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7-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(2S,4R)-4-(3,4-difluorobenzamido)-N-[2-(phenylamino)ethyl]pyrrolidine-2-carboxamide
2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-N-(propan-2-yl)pyrimidin-4-amine
7-[2-(benzyloxy)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-[2-(propan-2-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.5]undecane
(3S)-3-benzyl-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-one
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
3-chloro-4-({4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}methyl)phenol
3-(azocane-1-carbonyl)-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
2-ethyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)pyrimidine-5-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pent-4-enamide
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-(1-hydroxybutan-2-yl)-4-(hydroxymethyl)-N-[(2-methylphenyl)methyl]benzamide
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
5-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-N,N-dimethylpyrimidin-2-amine
N-{1-[1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-[4-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-6-methylpyrimidin-2-yl]phenol
2-({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
3-[1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-4-{3-methyl-6-oxo-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}benzene-1-sulfonamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
1-(6-methoxypyridin-3-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
(4aR,7aS)-1-ethyl-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(3-methoxyphenyl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-hydroxyphenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
methyl (2S,4R)-1-[3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanoyl]-4-hydroxypyrrolidine-2-carboxylate
5-chloro-4-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-dimethyl-1H-pyrazole
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
1-(adamantan-2-yl)-4-(2-methoxyethyl)-1,4-diazepan-5-one
N-[(2,6-dimethylpyridin-4-yl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
N-[(3S,4R)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-[2-(furan-2-yl)phenyl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
4-(1,3-benzothiazol-2-yl)-1-(pyridin-3-ylmethyl)piperazine-2-carboxylic acid
2,8-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
1-methyl-1'-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(1H-pyrazol-1-yl)-1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one
4-(4-methoxy-3,5-dimethylphenyl)pyridine
2-{4-[2-(3-methoxypropyl)piperidin-1-yl]quinazolin-2-yl}ethan-1-amine
8-(3-aminopropanoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
8-({3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
3,5-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2-oxazole-4-sulfonamide
(3aR,6aR)-2-methanesulfonyl-5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-(2-methoxyethyl)-4-(6-methylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(2-amino-2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
6-cyclopentanecarbonyl-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine