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2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(oxan-4-yl)acetamide
(3aS,6aS)-2-cyclohexyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-4-(propylsulfamoyl)-N-(pyrazin-2-ylmethyl)benzamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-phenyl-1,2-oxazole-3-carboxamide
1-[(3-methylthiophen-2-yl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-ethyl-N-(oxan-4-ylmethyl)-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
ethyl 2-(1-{[4-(4-acetyl-1,4-diazepan-1-yl)-8-methylquinazolin-2-yl]methyl}piperidin-2-yl)acetate
6-(1H-indol-3-ylmethyl)-3-[(E)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[4-(4-chlorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
(2S,4R)-N,N-diethyl-4-[5-(hydroxymethyl)furan-2-amido]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-[2-ethoxy-5-(trifluoromethyl)phenyl]urea
(3S,4R)-4-(3-fluorophenyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-(2H-1,3-benzodioxol-5-yl)-5-[1-(1H-imidazol-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
1-benzoyl-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}piperidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-4-sulfamoylbenzamide
8-[2-(2,6-dimethoxyphenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-[3-(2-methyl-4-phenylpiperazin-1-yl)-3-oxopropyl]methanesulfonamide
1-[2-({[3-(3-methylphenyl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-6-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)butan-1-one
N-(2-fluoroethyl)-3-{[1-(6-methylpyridin-2-yl)propan-2-yl]sulfamoyl}benzamide
3-(1H-pyrazol-1-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}benzamide
4-(5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazine-1-carbaldehyde
2-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
1'-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(2,2-diphenylcyclopropyl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2S)-pyrrolidine-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
propan-2-yl 4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-methyl-4-phenyl-9-[2-(pyridin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-[(2-methylphenyl)methyl]acetamide
5-(2-acetylbenzoyl)-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-chloro-N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(furan-2-yl)ethyl]amine
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(4-chlorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
1-[(2,5-dimethoxyphenyl)methyl]-3-(3-methoxybenzoyl)piperidine
1-(3-fluorobenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-5-methoxypyrimidine
1-[8-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
ethyl 1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]{[2-(morpholin-4-yl)pyridin-3-yl]methyl}amine