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2-(cyclohex-1-en-1-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]acetamide
5-(1-acetylpyrrolidin-2-yl)-N-[2-(cyclohex-1-en-1-yl)ethyl]thiophene-2-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2S)-3-(4-hydroxyphenyl)-2-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamido)propanamide
2-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-N-(4-fluoro-2-methylphenyl)acetamide
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-2-methyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-propylpyrimidine-5-carboxamide
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(5-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)benzamide
ethyl 2-(4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-[3-(3-fluorophenyl)phenyl]-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-4-carboxamide
4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-methyl-6-(propan-2-yl)pyrimidine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-[(4-ethylpiperazin-1-yl)methyl]-N,N-bis(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-(4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
N,2,6-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
9-(cyclopropylmethyl)-1-methyl-4-(2-methylfuran-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-4-(1H-pyrazol-1-yl)benzamide
3-(propan-2-yl)-5-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
3-(2H-1,3-benzodioxol-5-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-[2-(dimethylamino)ethyl]-N-ethyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1,2,3-thiadiazole-4-carboxamide
9-{[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
4-[3-(1H-imidazol-2-yl)benzoyl]-2-[(4-methoxyphenyl)methyl]morpholine
1-(2-methyl-1-benzofuran-7-carbonyl)-4-phenylpiperidin-4-ol
1-[7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
N2-cyclopropyl-N4-methyl-N4-[3-(oxolan-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-ethoxy-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3-{[1-(1-benzoylpiperidin-4-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-chloro-4-({[(5-ethylpyridin-2-yl)methyl](methyl)carbamoyl}amino)-N,N-dimethylbenzamide
N-propyl-4-(4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-(4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)ethan-1-one
methyl (1R,3S,3aR,6aS)-1-(2-methoxy-2-oxoethyl)-5-methyl-3-(6-methylpyridin-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(pyridin-3-yloxy)ethan-1-one
N-[(4-methylphenyl)methyl]-1-[2-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxamide
8-(1H-indol-2-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](furan-2-ylmethyl)(prop-2-en-1-yl)amine
1-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(2S,4R)-4-[(3-cyanopyridin-2-yl)amino]-1-(1H-indol-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
N-ethyl-5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrimidin-2-amine
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one