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6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one
3-{[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}propane-1,2-diol
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
(3R,4S)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
5-[2-(methylsulfanyl)phenoxymethyl]-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
1-{3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-oxopropyl}azepan-2-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[4-(3-fluorophenyl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-tert-butyl-4-(quinolin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
4-(benzyloxy)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
5,8-difluoro-2-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline
N-(adamantan-1-yl)-2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
N-(4-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)acetamide
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}ethan-1-one
1-[4-(3-methylpiperidine-1-carbonyl)phenyl]-3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]urea
{4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]morpholin-3-yl}methanol
1-(pyridin-2-yl)-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N4,5-dimethylpyrimidine-2,4-diamine
(3R,5S)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(3-methylphenyl)-5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}pyrimidine
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxo-N-(1,3-thiazol-2-yl)acetamide
N-cyclopentyl-2-(2-cyclopropylpyrimidin-5-yl)-6-fluoroquinoline-4-carboxamide
1-(cyclopropylmethyl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2,3,5,6-tetramethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
methyl[(6-methylquinolin-5-yl)methyl](pyrazin-2-ylmethyl)amine
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-1-methyl-1H-imidazole-4-sulfonamide
1-[3-(methylsulfanyl)propyl]-4-(1H-pyrrole-2-carbonyl)piperazine
4-(5-acetylthiophene-3-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
benzyl({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
(2R,3R,6R)-5-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(4-cyclopropanecarbonyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[1-(propan-2-yl)piperidine-3-carbonyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
6-methoxy-3-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1-benzofuran-2-carboxamide
2-(2-propoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-({5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine