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7-amino-4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(3-hydroxypropyl)-N-(propan-2-yl)acetamide
2-butyl-5-chloro-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1H-imidazole
N-[2-({2-[(3-chlorophenyl)methyl]-1,3-benzoxazol-6-yl}formamido)ethyl]acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-(2-methoxyethyl)-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-chloro-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzene-1-sulfonamide
3-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
methyl 3-(furan-3-amido)-5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[2-methoxy-5-(propan-2-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-1,2,5-thiadiazole-3-carboxamide
(2R,3R,6R)-3-phenyl-5-(2-propyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(oxolan-3-yl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazole
4-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
2-[(4-methylphenyl)methyl]-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
3,4-dichloro-N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
N-(cyclohexylmethyl)-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridine
1-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
8-chloro-3-[(2R)-pyrrolidin-2-ylmethyl]-3,4-dihydroquinazolin-4-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)acetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-phenylpropan-1-one
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
(4aS,7aR)-1-[2-(1H-indol-3-yl)ethyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
(3R,4R)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
5-(3-methoxyphenyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
1-({5-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-(3-fluorophenoxy)-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
4-{[1-(3-fluoro-4-methylbenzoyl)piperidin-3-yl]methyl}benzoic acid
N-(1-{[(furan-2-ylmethyl)(prop-2-yn-1-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
9-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
8-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoline
2-{1-[(2-ethoxyphenyl)methyl]-4-[1-(2-fluorophenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-[(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-5-methyl-2,3-dihydro-1H-indol-2-one
2-benzyl-8-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
[5-({[(3-chlorophenyl)methyl](cyclopropyl)amino}methyl)furan-2-yl]methanol
2-(2-aminoethyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylquinazolin-4-amine
(2S,4S)-4-amino-N-[(2-fluorophenyl)methyl]-1-methyl-N-propylpyrrolidine-2-carboxamide
1-(3,5-difluoropyridine-2-carbonyl)-4-(2-methoxybenzoyl)piperazine
4-chloro-3-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}-N-propylbenzamide
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N4-methyl-N4-[(4-methyl-1H-imidazol-2-yl)methyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
N-benzyl-N-methyl-3-({[3-(methylsulfanyl)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-[1-(dimethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol