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3-[(2-fluoro-4-methoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-methyl-N-{2-[1-(oxan-4-yl)piperidin-3-yl]ethyl}pyridine-3-carboxamide
ethyl 1-[2-(dimethylamino)ethyl]-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(3,4-dimethoxyphenyl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
1-[4-(3-acetylphenyl)phenyl]-3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
N-(1-hydroxy-2-methylpropan-2-yl)-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-{3-[3-(morpholine-4-carbonyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2,8-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]quinoline-4-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-(azepane-1-carbonyl)-N,1-dimethyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(1H-imidazol-1-yl)-1-(pyridine-3-sulfonyl)piperidine-4-carboxylic acid
N-tert-butyl-2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylformamido)acetamide
(2S,4S)-4-[2-(3-chloro-4-fluorophenoxy)acetamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
(4aS,7aR)-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(but-3-enoyl)-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-3-(1,2-oxazinan-2-yl)propanamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine-1-carboxamide
N,N-dimethyl-2-{[3-(4-methylphenyl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-{5-[1-(1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}-1,4-oxazepane
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-1-phenyl-1H-pyrazole-4-carboxamide
(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-(naphthalene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]-2-ethyl-1H-1,3-benzodiazole
3,5-dimethyl-1-{1-[(5-propylfuran-2-yl)methyl]azetidin-3-yl}-1H-pyrazole
(3S,4R)-4-(pyridin-3-yl)-1-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidine-3-carboxylic acid
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(4-methylpiperazin-1-yl)butyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
4-(5-benzyl-4-cyclopropanecarbonyl-2-oxopiperazin-1-yl)benzonitrile
5-{1-ethyl-2,7-dioxo-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinolin-9-yl}thiophene-2-carboxylic acid
[(1-cyclopentylpiperidin-4-yl)methyl][(4-methoxy-2,3-dimethylphenyl)methyl](pyridin-3-ylmethyl)amine
1-(3-methoxyphenyl)-4-[(1-methyl-1H-indol-6-yl)methyl]piperazin-2-one
7-chloro-3-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
2-{[(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-(1H-imidazol-4-yl)-1-[2-(4-methoxyphenyl)phenyl]-1H-imidazole
1-(3-fluorophenyl)-3-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-benzoyl-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazine
3-(2-methoxyethyl)-1-(3-methylphenyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-(2-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}ethyl)acetamide
4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(1H-1,3-benzodiazol-2-ylmethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[4-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)phenyl]acetamide
2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-butyl-4-ethyl-1-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide