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2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-methylacetamide
3-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}-N-[(2R)-pyrrolidin-2-ylmethyl]benzamide
dimethyl({5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}methyl)amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methylphenoxy)ethan-1-one
{3-ethyl-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}methanol
N-[(2-fluorophenyl)methyl]-2-{[3-(pyrrolidin-1-yl)propyl]amino}acetamide
2-(3-{1-[(5-chlorothiophen-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4-oxazepane
4-[3-(azepan-1-yl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
1-[(3-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
1-methanesulfonyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
4-(7-fluoro-2-methylquinoline-4-carbonyl)-3-methyl-1-phenylpiperazin-2-one
N-[3-(1H-imidazol-1-yl)propyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-{[3-(methylsulfanyl)phenyl]methyl}-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(propan-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-hydroxy-4-(pyridin-3-yl)-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
2-(1-benzofuran-2-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(2,3-difluoro-4-methoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-methyl-14-(5-methyl-1-propyl-1H-pyrazol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(5-methylpyrazin-2-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
4-(3-fluorophenoxy)-1-[4-(piperidin-3-yl)benzoyl]piperidine
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N,8-dimethyl-N-(oxan-4-yl)quinoline-4-carboxamide
4-(5-methylpyrazine-2-carbonyl)-2-(naphthalen-1-ylmethyl)morpholine
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-[1-(methylsulfanyl)propan-2-yl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[(dimethylamino)methyl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]azepan-4-ol
1-ethyl-3,5-dimethyl-4-({2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1H-pyrazole
4-(4-ethoxypiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(1H-1,3-benzodiazol-2-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
N,N-dimethyl-6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]pyrazin-2-amine
(2S,4R)-4-amino-N-ethyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
4-(hydroxymethyl)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}azepan-4-ol
(1R,5R)-N,N-dimethyl-6-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
7-fluoro-2-methyl-3-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-(3,4-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
8-[(2R)-2-amino-3-methoxypropanoyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidin-3-yl)methyl]benzamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
3-(3-methyl-1-propyl-1H-1,2,4-triazol-5-yl)benzoic acid
2-{[(3R,5S)-1-benzyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
2-(3-hydroxypropyl)-9-{[4-(propan-2-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-5,8-dimethyl-1,4-dihydroquinolin-4-one
4-chloro-1-methyl-3-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-1H-indazole