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5-[methyl(1,2-oxazol-3-ylmethyl)amino]-1-[(4-methylphenyl)methyl]azepan-2-one
N-[2-(2-chlorophenyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
1-(furan-3-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
[4-(3-phenylpropyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl]methanol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(pyrazin-2-yl)ethyl]benzamide
7-methyl-2-[4-(pyrrolidin-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
2,6-dimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]quinoline-4-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
(4aS,7aR)-1-[3-(1H-pyrazol-1-yl)propanoyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-methoxyethyl)-2-[1-(4-methoxyphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
5-({[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)-N-methylfuran-2-carboxamide
4-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
4-(pyrrolidine-1-carbonyl)-1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)piperidine
5-methyl-N-{2-[(4-methyl-1,2,3-thiadiazol-5-yl)sulfanyl]ethyl}-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2-(trifluoromethyl)morpholine
2-({[4-(2-aminoethyl)phenyl]methyl}(cyclohexyl)amino)ethan-1-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-propylpyrimidine-5-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
5-(2,4,6-trifluorophenoxy)-1-azabicyclo[3.2.1]octane
7-(1,4-dioxane-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-4-(hydroxymethyl)-1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-ol
4-chloro-1,5-dimethyl-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-3-carboxamide
2-ethyl-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1-(propan-2-yl)piperazine
1-(3-fluorophenyl)-3-{1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
8-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3R,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}pyridine
4-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-butyl-1-methylpiperazin-2-one
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-(1-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1'-[2-(2-methoxyethoxy)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-[2-(3-fluorophenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-methyl-4-(1-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}ethyl)piperazine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-(pyrrolidin-1-ylmethyl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
2-methoxy-1-{4-[1-(pent-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]piperidin-1-yl}ethan-1-one
4-[4-(3-ethylpiperazin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
5,6-dimethyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[1-(1H-indol-5-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(1R,3S)-3-methoxy-7-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}-7-azaspiro[3.5]nonan-1-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-[5-(cyclopropylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(3-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
1-methyl-2-(morpholin-4-yl)-N-[2-(pyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
(3aS,6aS)-2-methyl-5-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(1H-pyrazol-1-yl)benzoyl]-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine