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5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridine-2-carbonitrile
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1H-pyrazole-4-carboxamide
(3aR,6aR)-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(cyclopentylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-(1H-1,3-benzodiazol-2-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-chloro-N,N-dimethyl-3-phenyl-1H-indole-2-carboxamide
1-(4-cyclopentylpyrimidin-2-yl)-N,N-diethylpyrrolidin-3-amine
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}propan-1-one
1-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}azepan-2-one
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-hydroxy-4-methylpentan-1-one
methyl (2S)-1-(2-{4-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}acetyl)pyrrolidine-2-carboxylate
1-(2,3-dihydro-1H-inden-2-yl)-N-(furan-2-ylmethyl)piperidin-3-amine
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(1,2-oxazolidin-2-yl)propanamide
4-[2-(butylsulfanyl)pyrimidin-5-yl]-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
7-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
7-fluoro-N,3-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
N,N-dimethyl-3-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}propanamide
methyl 4-(4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]piperazine-1-carboxamide
2,3-dimethoxy-N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
methyl 2-{8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
7-(3-chlorophenyl)-4-(furan-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
dimethyl[3-(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
1-{2-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-pyrazole
3-(2-butoxyacetamido)-4-(2-methylpiperidin-1-yl)benzamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-N-(3-methoxypropyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{2-[1-(2-propoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
8-fluoro-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}quinoline
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-2-(thiophen-3-yl)ethan-1-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}diethylamine
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(3-cyano-4-methoxyphenyl)-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-chloro-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-5-(trifluoromethyl)benzamide
2-(4-fluoro-3-methylphenyl)-2-[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]acetic acid
4-(2,3-dihydro-1H-indene-1-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-({4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]piperidin-4-ol
3-(4-methoxy-3,5-dimethylbenzoyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
2-(azepan-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[3-(2-chlorophenoxy)propyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
(4aS,8aR)-1-(2-aminoethyl)-6-(quinoline-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-6-oxo-1,6-dihydropyridine-2-carboxamide