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6-(4-methoxy-2,6-dimethylphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[1-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-(1H-pyrazol-4-yl)pyridine
2-{1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}pyridine
(1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
3-{[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl}-7-methylquinolin-2-ol
1-{1,3-dioxo-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]-2-(5-fluoro-2-methylphenyl)acetic acid
1-(2,2-dimethylpropyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
1-(3-ethyl-1H-pyrazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{imidazo[1,2-a]pyridin-3-yl}-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
1-(4-methyl-1H-pyrrole-2-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
4-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl}benzoic acid
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetamide
3-[2-(1H-indol-6-yl)ethyl]-1λ6-thiolane-1,1-dione
N-[1-(3-methylpyridin-2-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
2-ethoxy-6-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
3-(4-chlorophenyl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
4-phenoxy-1-[2-(pyrrolidin-1-yl)propanoyl]piperidine-4-carboxylic acid
N-[2-(3-methoxyphenyl)-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
(1S,5R)-3-(4-aminopyrimidin-2-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(3-phenylpropyl)morpholin-4-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(2S,4S)-4-acetamido-N-ethyl-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxamide
2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
(2S,4S)-1-(3-phenylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
1-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
4-chloro-1-[5-(morpholine-4-carbonyl)furan-2-yl]-1H-indazole
3-methanesulfonamido-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
9-[2-(methylsulfanyl)pyrimidin-4-yl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-{1-[3-(piperidin-4-ylmethyl)benzoyl]piperidin-4-yl}phenol
N-[2-(4-phenylpiperidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
1-ethyl-4-({3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperazine
N-ethyl-N-methyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-chloro-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-5-(trifluoromethyl)benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})(quinolin-8-ylmethyl)amine
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
9-[(4-hydroxyphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-amino-6-{4-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
{1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropyl}methanol
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]thiomorpholine-4-carboxamide
N-(6-methylpyridazin-3-yl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide