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3-[(2,4-dimethylphenyl)methyl]-1λ6-thiane-1,1-dione
1-[2-(dimethylamino)-4-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-[(4-fluorophenyl)formamido]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[(2-fluorophenyl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
3-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-5-(4-methylpiperidine-1-carbonyl)-1,4-dihydropyridin-4-one
4-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-2-one
N-[2-(benzylsulfanyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-(methoxymethyl)-N-[3-(2-phenylacetamido)phenyl]furan-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
5-(methoxymethyl)-N-[2-(piperidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[3-(4-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
1-[3-({[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}amino)propyl]pyrrolidin-2-one
2-(dimethylamino)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(3-methylphenyl)acetamide
5-(4-benzoylpiperidine-1-carbonyl)-1-[(2-fluorophenyl)methyl]piperidin-2-one
2-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
3-({[2-(2-phenoxyphenyl)ethyl]amino}methyl)piperidin-3-ol
(1R,2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-propylcyclopropane-1-carboxamide
(2S)-N1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}propane-1,2-diamine
(3S,4S)-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
8-[4-(4-chlorophenyl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-(4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
N'-(3-chloro-4-methylphenyl)-N-[3-(propan-2-yloxy)propyl]propanediamide
3-{5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(3-{1-[3-(dimethylamino)propyl]-1H-pyrazol-3-yl}phenyl)benzonitrile
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,6-dimethyl-N-[3-(4-methylbenzenesulfonamido)propyl]pyrimidine-4-carboxamide
3-chloro-N-[1-(thiophen-2-yl)ethyl]pyridine-4-carboxamide
3-(3-fluorophenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrazine-2-carboxylic acid
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-4-methylbenzamide
1-{5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
2-[2-(azocan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylacetamide
2-methyl-N-({3-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
5-(2,6-dimethylphenyl)-2,4-dimethoxypyrimidine
(3S,4S)-1-(6-methyl-2-propylpyrimidin-4-yl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
3-(2-methoxyethyl)-1-[3-(piperazin-1-yl)propanoyl]piperidine-3-carboxylic acid
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
3-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-ol
1-(oxan-4-yl)-N-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
4-(1-methylpyrrolidin-3-yl)piperidine
2-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
2-ethoxy-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylpyridine-3-carboxamide
N,3-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide