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1-(3-{[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propyl)pyrrolidin-2-one
3-cyclohexyl-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[1-(2-hydroxyethyl)-5-[(1S,2R)-2-(pyrrolidine-1-carbonyl)cyclohexyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
2-cyclopropyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
6-cyclopentyl-N-(1,4-dioxan-2-ylmethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetic acid
N-cyclooctyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-ethyl-N-(1-hydroxybutan-2-yl)-5-methyl-N-(thiophen-2-ylmethyl)thiophene-3-carboxamide
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-3-carbonitrile
15-methyl-12-(piperidine-1-carbonyl)-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-(1,3-oxazole-5-carbonyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-[(5-chloro-2-propoxyphenyl)methyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
N-benzyl-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N,2,8-trimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]quinoline-4-carboxamide
1-(azepan-1-yl)-3-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]propan-2-ol
N-(1-{[(1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-3-carboxamide
4-(2-chlorophenyl)-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(2-chlorobenzoyl)-3-(3-fluoro-4-methoxybenzoyl)piperidine
8-(2,1,3-benzothiadiazol-4-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-(naphthalen-2-yloxy)-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
(3S)-4-(1-benzothiophene-5-carbonyl)-3-ethylmorpholine
naphthalen-1-yl (7R,9aR)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[3-(2-phenylethyl)piperidin-1-yl]-3-(piperidine-1-carbonyl)pyridine
N-methyl-3-(1-methylpiperidin-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
1-{1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}-2-phenylethan-1-ol
1-(2-methylphenyl)-4-[2-(prop-2-en-1-yloxy)benzoyl]piperazin-2-one
2-[2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetamide
(1r,4r)-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4-methylcyclohexane-1-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
1,3-dimethyl-5-({[1-(2-methylpropyl)piperidin-4-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}urea
5-(1-benzofuran-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,2,4-triazin-3-amine
(1S,3R)-3-amino-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)cyclopentane-1-carboxamide
N-(2-methoxyethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-2-ylmethyl)propanamide
1-(2-methylpyridin-4-yl)-4-[3-(trifluoromethyl)benzoyl]-1,4-diazepane
2-(oxolan-2-ylmethyl)-9-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-{5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}piperidine