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1-{5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
3-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N-(2-chloro-4-fluoro-5-methylphenyl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
2-(4-cyclopentylpyrimidin-2-yl)benzoic acid
1-[4-(1H-imidazol-1-yl)butanoyl]-1,4-diazepane-6-carboxylic acid
4-(hydroxymethyl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-ol
4-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-chlorophenyl)morpholine
N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
1-{2-[2-(5-acetylthiophen-3-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-[1-(pyrimidin-4-ylmethyl)-1H-imidazol-2-yl]-1H-1,3-benzodiazole
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
2-[1-(1-methylpiperidin-4-yl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
7-methyl-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-dihydroquinolin-2-one
4-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}piperazine-2-carboxylic acid
N-methyl-N-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)acetamide
ethyl 5-[({1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidin-3-yl}formamido)methyl]furan-2-carboxylate
6-[(2-hydroxyethyl)(methyl)amino]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
3-[(3R,4S)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-(1,4-dimethylpiperazin-2-yl)-1-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}ethan-1-one
[(2-ethylpyrimidin-4-yl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
(4aR,7aS)-1-acetyl-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-butyl-1-(3-methylphenyl)-4-(1,2-oxazole-3-carbonyl)piperazin-2-one
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}imidazo[1,2-a]pyrimidine-2-carboxamide
3-(1H-indol-5-yl)-1-methyl-1-(thian-4-yl)urea
{1-[4-(4-propylphenyl)benzoyl]pyrrolidin-3-yl}methanamine
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-4-(pyridin-3-yl)piperazine
(benzylsulfamoyl)({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)amine
8-benzyl-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-5-{1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(1-benzofuran-2-yl)-1-(oxan-4-yl)-1H-imidazole
1-(propan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
N-ethyl-3-(3-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
1-(2-methoxyphenyl)-4-(5-propyl-1,2-oxazole-4-carbonyl)piperazin-2-one
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,5-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(ethylsulfanyl)-5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)pyrimidine
3-(3-fluoro-4-methoxybenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
1-[(4,5-dimethylfuran-2-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(4S,4aS,8aS)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-1-methylpiperazine-2-carboxylic acid
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(trifluoromethyl)pyrimidin-2-amine
3-[(propan-2-yl)(3,3,3-trifluoropropyl)amino]propanamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
13-[3-(1H-pyrazol-1-ylmethyl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one