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7-chloro-3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-ethyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-3-hydroxypyridine-2-carboxamide
3,3-dimethyl-1-({5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,2-oxazole-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(5-tert-butyl-1H-pyrazol-3-yl)methyl]amine
N,2,6-trimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]quinoline-4-carboxamide
2-(4-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
5-hydroxy-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrazine-2-carboxamide
4,6-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-2-amine
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
N-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}methanesulfonamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
(2-methoxy-5-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}phenyl)methanol
1-cyclohexyl-3-(cyclopropylmethyl)-N-(1,2-oxazol-3-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methanesulfonyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(3E)-1-(2-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)pent-3-en-1-one
1-(4-cyclohexylphenyl)-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
N-[3-(1,3-thiazol-4-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
4-(1-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
({4-ethyl-5-[1-(5-ethylthiophene-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
1-ethyl-4-[(2S)-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N'-cyclohexyl-N-(2-methylphenyl)-N'-(pyridin-2-ylmethyl)propanediamide
1-{1-[(2-hydroxy-7-methylquinolin-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
1-methyl-3-(piperidine-1-carbonyl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(3S,4S)-1-(2-phenylmethanesulfonylbenzoyl)piperidine-3,4-diol
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-hydroxyethan-1-one
(3S)-1-[2-(2,5,7-trimethyl-1H-indol-3-yl)ethyl]pyrrolidin-3-ol
7-(3-{[2-(methylsulfanyl)phenyl]carbamoyl}propanoyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-(2-methoxyethyl)-1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]piperidine-3-carboxylic acid
4-(azepan-1-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]-4-oxobutanamide
2-{4-[4-(2-methylpropyl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
N-({1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
5-ethyl-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-4-amine
3-{[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
(1S,2R)-N1-(2,1,3-benzoxadiazol-5-ylmethyl)-N2-butylcyclohexane-1,2-dicarboxamide
(3R,4R)-4-[(8-methoxyquinolin-2-yl)amino]piperidin-3-ol
1-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
{1-[2-(4-fluorophenoxy)ethanesulfonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-[2-methyl-4-(pyridin-4-yl)phenyl]pyridine-3-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]pyrimidin-2-amine
(3R,4R)-1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
N-(adamantan-2-yl)-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2,7-dimethyl-N-[2-(4-sulfamoylphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxamide