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(3S,4S)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
3-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
(4aS,7aR)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(1H-pyrazol-5-ylmethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-(pyrimidin-2-yl)-N-(quinolin-8-ylmethyl)piperidin-3-amine
(2S,4R)-4-(cycloheptylamino)-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-4-carboxylate
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-[(3-methylphenyl)(thiophen-2-yl)methyl]acetamide
4-(piperidin-3-ylmethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-methyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-oxaspiro[4.4]nonane-4-carboxamide
5-(2,3-dimethoxyphenyl)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazole
N-cyclohexyl-2-cyclopropyl-N-[(4-fluorophenyl)methyl]pyrimidine-5-carboxamide
1-{1-[(3-chlorophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[(1-ethylpyrrolidin-3-yl)methyl]-4-methyl-1,3-benzothiazole-6-carboxamide
[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
methyl 4-{2-amino-3-cyano-7-methyl-5H,7H-thieno[3,4-b]pyridin-4-yl}-1H-pyrazole-3-carboxylate
2-methyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(2E)-3-phenylprop-2-enoyl]pyrrolidin-3-yl]acetamide
2-ethyl-4-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)pyrimidine
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]acetamide
3-(2-ethoxyethyl)-1-[(4-methoxypyridin-2-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-{2-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(thiolan-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-[(3-phenoxyphenyl)methyl]pyrrolidine-2-carboxamide
(2S,3S)-3-methyl-2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}pentanamide
N-(2-methanesulfonamidoethyl)quinoxaline-5-carboxamide
3-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-{[(1-benzofuran-2-ylmethyl)amino]methyl}-N,N-diethylpyridin-2-amine
1-(4-chlorophenyl)-N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]cyclopropane-1-carboxamide
N-(2-methoxyethyl)-2-(2-methyl-5-oxopyrrolidin-1-yl)-N-(naphthalen-1-ylmethyl)acetamide
1-cycloheptyl-N-(1H-imidazol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-cyclopropylethyl)-1,3-oxazole-4-carboxamide
N-[(2,4-dihydroxyphenyl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)acetamide
7-methyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-[3-(2-methyl-1H-imidazol-4-yl)benzoyl]piperidine
1-(3-chlorothiophene-2-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
3-[4-(ethoxycarbonyl)-4-(3-phenylpropyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
1-(2,3-dihydroxypropyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
4-{[1-(2-fluoro-6-methoxybenzoyl)piperidin-3-yl]methyl}benzoic acid
2-{[5-(1H-indol-3-ylmethyl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(pyrazin-2-yl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
9-[4-(aminomethyl)benzoyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[3-(2-fluorophenyl)pyrrolidin-1-yl]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
N'-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}ethanediamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[1-(propan-2-yl)piperidine-3-carbonyl]piperidine