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4-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
3-[5-({2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyridine
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-1-(oxolane-2-carbonyl)piperidin-4-amine
9-(3-hydroxy-4-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
3-[(3-hydroxyazetidin-1-yl)methyl]-7-methyl-1,2-dihydroquinolin-2-one
1-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-5-methoxyfuran-2-carboxamide
2,7-bis(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-fluoro-4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
N-benzyl-2-(1H-pyrazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)butanamide
5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
(1S,4S)-5-[2-(2-chlorophenyl)acetyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
{4-[3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]phenyl}methanamine
6-{[1-(4-fluorophenyl)propan-2-yl]amino}-2-methylheptan-2-ol
2-{2-[(1R,5S)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
N-{2-[methyl(phenyl)amino]ethyl}-1-propanoylpiperidine-3-carboxamide
4-({[5-(methoxymethyl)furan-2-yl]methyl}amino)-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(1R,3S,4S)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carboxamide
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(methylsulfanyl)pyridine-3-carboxamide
N-[4-(pyrimidin-5-yl)phenyl]butanamide
ethyl 2-{[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}acetate
1-{furo[3,2-c]pyridin-4-yl}-3-(2-phenoxyethyl)piperidine-3-carboxylic acid
3-[(2-methyl-1,3-oxazol-4-yl)methyl]-5-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-methyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-amine
(3aS,6aS)-2-(ethanesulfonyl)-5-(1H-indol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[5-(ethylcarbamoyl)-2-methylphenyl]pyrrolidine-1-carboxamide
5-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
(4-{[4-(2-chloro-6-fluoro-3-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
N-[2-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-2-yl)ethyl]acetamide
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
3-({2-[1-(5-fluoro-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-({5-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
(3R,4R)-4-amino-1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-3-ol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-(5-ethyl-2-methylpyrimidin-4-yl)-1λ6-thiomorpholine-1,1-dione
2,4-dimethoxy-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1,3,5-triazine
(4aS,7aR)-1-(3,3-dimethylbutyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(3-methylphenoxy)azetidin-1-yl]propan-1-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3,4-difluorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
5-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-N-methylpyrimidin-2-amine