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6-methoxy-1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(2-fluorophenyl)-3-phenylpropanamide
8-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(3R,4S)-4-cyclopropyl-1-[2-(methylcarbamoyl)ethyl]pyrrolidin-3-yl]-4-(methoxymethyl)benzamide
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
3-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-N-[2-(dimethylamino)ethyl]propanamide
1-[(4-fluorophenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepane
2-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-2-yl}pyridine
4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-phenylpiperazin-2-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(methylamino)-N-(propan-2-yl)pyridine-4-carboxamide
1-(1,2-oxazol-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3,5-dichloro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N,4-dimethylbenzamide
methyl[3-(1H-pyrazol-1-yl)propyl](thiophen-3-ylmethyl)amine
2-chloro-5-acetamido-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}benzamide
2,6,8-trimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
5-methoxy-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,4-dihydropyridin-4-one
1-methyl-3-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2-dihydroquinolin-2-one
1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
N-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1-ethyl-1H-indole-5-carbonyl)pyrrolidin-3-yl]methanol
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(quinolin-2-yl)pyrrolidin-3-yl]methanol
5-benzamido-1-cyclopentyl-N-[2-(furan-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-[(2-hydroxyethyl)({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
(3R,4R)-1-[(5-chlorothiophen-2-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-methyl-4-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}phenol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1'-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3H-spiro[2-benzofuran-1,4'-piperidine]-3-one
N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}pyridine-3-carboxamide
4-methyl-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyrimidin-2-amine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-imidazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methylacetamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
ethyl 2-(2,4-dimethoxyphenyl)pyridine-3-carboxylate
3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridin-2-ol
1-cyclopentyl-4-[({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
2-[1-(cyclohexylmethyl)-4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-cyclobutyl-3-{[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)sulfamoyl}benzamide
3-ethyl-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]urea
2-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]-N-methylpyridine-3-carboxamide
ethyl 1-{[3-(methylsulfanyl)phenyl]carbamoyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-(4-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenyl)-2-methylbutan-2-ol
4-(2-{[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(trifluoromethyl)benzamide
4-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole
2-(4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
(2E)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(3,4-dimethoxyphenyl)prop-2-en-1-one
2-(hydroxymethyl)-N-[4-(trifluoromethyl)phenyl]azepane-1-carboxamide