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4-[(2-methylpyridin-3-yl)oxy]-1-(1,2-oxazole-3-carbonyl)piperidine-4-carboxylic acid
(3S,7S,8aS)-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
6-({3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(1-methylpyrrolidin-2-yl)acetamide
1-[(4-fluorophenyl)methyl]-4-(5-methylpyrazine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-[2-(4-chlorophenyl)ethyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-({[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(2,4-dichlorophenoxy)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
(1R,3S)-7-(dimethyl-1,3-thiazole-5-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1H-indol-5-yl)methyl]acetamide
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
[(2-fluorophenyl)methyl](methyl){[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-methyl-1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}urea
3-(4-methoxyphenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
(3S,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(propan-2-yl)piperidine-3-carboxamide
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-(thiophene-2-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-methylacetamide
(2S)-3-(4-hydroxyphenyl)-2-({6-methylpyrazolo[1,5-a]pyrimidin-3-yl}formamido)propanamide
N-[4-methyl-3-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
7-(cyclopropylmethyl)-2-[3-(2-fluorophenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(3-fluorophenyl)-3-{1-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}pyrimidine
6-[(oxolan-2-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
(1S,5R)-6-(cyclobutylmethyl)-3-[(2,4-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-chloro-4,5-difluorophenyl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
3-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,2-dihydroquinolin-2-one
2-{[4-(3-chlorophenyl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(1-benzylpiperidin-4-yl)ethyl]amine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
2-{3-[hydroxy(phenyl)methyl]-5-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-{2-[2-(6-chloro-2-fluoro-3-methylphenyl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
(3aR,5S,6S,7aS)-2-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)-octahydro-1H-isoindole-5,6-diol
3-cyclopropyl-5-(oxolan-3-ylmethyl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-(thiophen-3-yl)propan-1-one
1-{4-[(3-ethenylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methoxypropan-1-one
2-(1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidin-2-yl)-1,3-thiazole
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol
N-(4-methoxy-2-methylphenyl)-3-[1-(5-phenylpentanoyl)piperidin-3-yl]propanamide
N3-tert-butyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrimidin-2-amine
7-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(3R,5S)-1-(furan-2-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1-methyl-1H-imidazole-2-carboxamide
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
3-(furan-2-yl)-2-(4,5,6,7-tetrahydro-1-benzothiophen-2-ylformamido)propanoic acid