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{2-[2-(1-cyclohexanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
1-{4-[2-(4-fluorophenyl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1,5-dimethyl-4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-methyl-N-[2-(2,3,6-trimethylphenoxy)ethyl]pyrazine-2-carboxamide
4,6-dimethyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(pyrazin-2-yl)-1,4-diazepan-5-one
(1S,5R)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2,6-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidine-4-carboxamide
(1R,5S,6R)-3-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-N-[2-(1H-imidazol-1-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2,6-dimethyl-4-(1-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-imidazol-2-yl)phenol
1-(2-methoxyethyl)-3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-[(5-methylthiophen-2-yl)methyl]urea
4-(5-ethyl-1,3,4-oxadiazol-2-yl)-1-phenylpiperazin-2-one
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]propanamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
3-[1-(2-cyclopropyl-1H-imidazol-1-yl)ethyl]-4-(2-methoxyethyl)-4H-1,2,4-triazole
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-2-(morpholin-4-yl)propanamide
4-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)benzoic acid
3-(2-fluoro-6-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-(cyclohexylmethyl)-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
1-cyclopropanecarbonyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(4S)-4-amino-5-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-5-oxopentanoic acid
1-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl}imidazolidin-2-one
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
2-(1H-imidazol-1-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
1-cyclopropyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5,6-dimethylpyrimidin-4-amine
1-ethyl-3,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-4-carboxamide
N-[4-(4,5,6-trimethylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
(1S,5R)-6-propyl-3-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-3,4-dimethyl-1-(4-propylbenzoyl)pyrrolidin-3-ol
2-{4-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
6-methoxy-1-methyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole
N-ethyl-2-[4-(1H-pyrazol-3-yl)phenyl]acetamide
6-methoxy-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]propan-1-one
1-ethyl-8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxylic acid
4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-one
6-methoxy-N-(2-methylpropyl)-2-oxo-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
(butan-2-yl)[(2E)-3-(furan-2-yl)prop-2-en-1-yl](pyridin-3-ylmethyl)amine
2-(1-cyclohexylpiperidin-4-yl)-N-methylacetamide
4-(2,5-dimethoxyphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H-1,2,4-triazole
2-{2-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
2-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(methylamino)acetamide
3-(propan-2-yl)-4-[1-(propan-2-yl)piperidin-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)-2,8-diazaspiro[4.5]decane