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1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidine-3-carbonitrile
4-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2,1,3-benzoxadiazole
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(azepan-1-yl)-3-[3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[(3R,4R)-4-hydroxypiperidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
methyl 4-oxo-4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}butanoate
N4,6-dimethyl-N4-[3-(oxolan-2-yl)propyl]pyrimidine-2,4-diamine
2-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-6-fluorobenzamide
N4-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-N2,6-dimethylpyrimidine-2,4-diamine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]acetamide
3-methoxy-1-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
4-ethyl-5-methyl-N-[1-(pyridin-2-yl)propyl]thiophene-3-carboxamide
3-(4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(3-hydroxy-3-phenylpyrrolidin-1-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
9-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
9-(2,3-difluorobenzoyl)-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1'-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[1-(thiophen-2-yl)butyl]propanamide
5-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane-1-carbaldehyde
4-{[4-(3,4-dimethylphenoxy)phenyl]methyl}piperazine-2-carboxylic acid
[(1R,3R,3aS,6aR)-5-ethyl-1-(2-methylpropyl)-3-[1-(propan-2-yl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(3aR,6aR)-2-cyclohexyl-5-(thiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(1H-pyrazol-3-yl)-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridine
1-{1-[6-(3-hydroxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-[2-(2-oxo-1,2-dihydropyridin-3-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
7-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[(2-chlorophenyl)methyl]-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-benzyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1H-1,2,4-triazole
8-(2-methylquinolin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(cyclopropylmethyl)-4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-2-(propan-2-yl)-1,4-diazepane
1-ethyl-5-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-2,3-dimethyl-N-(oxolan-2-ylmethyl)quinoxaline-6-carboxamide
2-cyclohexyl-N-(1,2-oxazol-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]-N,N-dimethylpyridin-2-amine
1'-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1,2-oxazinan-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
2-(2-hydroxyethyl)-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-4-methyl-N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)benzamide
4-(5-chloropyridine-3-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-(2-hydroxyethyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-1-(2-fluoro-4-methylphenyl)urea
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
3-(4-methoxyphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid