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2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1,3-thiazole-4-carboxamide
N-butyl-N,6-dimethyl-2-(morpholin-4-yl)pyrimidin-4-amine
5-{[3-(propan-2-yloxy)propyl]carbamoyl}-1H-imidazole-4-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-(isoquinolin-5-ylmethyl)-N-methylpropanamide
3-(but-2-yn-1-yl)-5-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-{[3-(furan-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one
N-[3-({[cyclopropyl(6-methylpyridin-2-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
[(3-methoxyphenyl)methyl](methyl){[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}amine
4-[(4-fluoro-2-methylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methoxy-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-{1-[({2-[4-(propan-2-yloxy)phenyl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}thiophene-3-carboxamide
3-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}propane-1,2-diol
2-[(1R,3S,3aS,6aR)-5-benzyl-1-(hydroxymethyl)-3-(2-methylphenyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
1-tert-butyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
1-{3-[4-(2,3-dimethoxyphenyl)-1H-1,2,3-triazol-1-yl]propyl}pyrrolidin-2-one
2-(methylsulfanyl)-5-(1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)pyrimidine
3-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-(ethanesulfonyl)-5-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(4-{[(2-methoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
2-(3-methoxyphenyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
N-{[4-(morpholin-4-yl)phenyl]methyl}-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,5-dimethyl-1H-pyrazole
5-amino-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1H-pyrazole-3-carboxamide
(1R,2R,6S,7S)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
(2H-1,3-benzodioxol-5-ylmethyl)[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](pyridin-3-ylmethyl)amine
4-methyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
N,5,6-trimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-methyl-4-{3-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane-1-carbaldehyde
2-(dimethylamino)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,4-dimethylpyrimidine-5-carboxamide
2-(2-oxopiperidin-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-(cyclohex-1-en-1-ylmethyl)-1-(2-methoxyacetyl)piperidine-4-carboxamide
(3R,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-ethylpiperidine-3,4-diol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(4-hydroxyphenyl)methyl]piperidine-4-carboxamide
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-(2-fluorophenyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-{2-[4-fluoro-3-(trifluoromethyl)phenyl]phenoxy}propanamide
3-{4-[(2,3-difluoro-4-methylphenyl)methyl]piperazin-1-yl}propanamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]pyrrolidin-3-ol
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1,2,4-oxadiazol-3-yl)piperidine
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4-methylpiperazine
(2S)-2-(hydroxymethyl)-N-(1H-indol-5-yl)pyrrolidine-1-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-ol