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2-methoxy-1-(1'-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
8-(oxolan-3-ylmethyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-butyl-4-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
3-{[3-methoxy-2-(prop-2-yn-1-yloxy)phenyl]methyl}-3,9-diazaspiro[5.5]undecane
(2-{4-[4-(azepan-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propyl)dimethylamine
(benzylsulfamoyl)({2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})amine
2-(4-ethylpiperazin-1-yl)-N-[(2-methylphenyl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 4-(2-phenoxyethyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
2,3-dimethyl-6-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]quinoxaline
4-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
N-[(2-chlorophenyl)methyl]-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-4-hydroxyquinoline-6-carboxamide
methyl({[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]methyl})(pyridin-3-ylmethyl)amine
5-{2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-(cyclopent-2-en-1-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopentan-1-ol
(2R,6R)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-(2-{[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-[(2S)-5-oxopyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl}acetic acid
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}morpholine-4-sulfonamide
2-ethyl-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]butan-1-one
1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-3-(1H-imidazol-1-ylmethyl)piperidine
4-[(5-{2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-[2-(trifluoromethyl)phenyl]ethan-1-ol
2-(dimethylamino)-1-{6-methyl-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidine-4-carboxylate
1-(4-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
8-(2-amino-6-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,9aR)-1-({[(5-methoxy-1H-indol-2-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-[(2,5-dimethylphenyl)methyl]-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
4-({5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}(methyl)amino)-2-methylbutan-2-ol
N-[3-(cyclohexyloxy)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-butanoyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N,2-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-chloro-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5-(1H-pyrazol-1-yl)benzamide
3-[1-(4-chlorobenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
(4aR,8aR)-7-[2-(3-fluorophenyl)ethyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-(2-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2,7-dioxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,3-diazepane-4-carboxamide
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
6-cyclopropyl-N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]pyrimidin-4-amine
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-(4-methoxyphenyl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
2-(2-{[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}phenoxy)acetic acid
4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane