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3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-chloro-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{3,5-dimethyl-4-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-amido]-1H-pyrazol-1-yl}acetic acid
4-{1-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-4-yl]ethyl}morpholine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylbutanamide
N-(3-chloro-4-fluorophenyl)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-{[(2,3-dimethoxyphenyl)methyl]amino}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
N-(2-methoxyethyl)-2-(pyridine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
2-(2,6-difluoro-3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-2-ylmethyl})amine
N-[(5-methylpyrazin-2-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
(4aS,8aR)-6-[(2-aminopyridin-3-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
6-(1-methylpiperidin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-4-amine
6-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
ethyl 1-(4-ethenylbenzoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-({5-[(2,3-difluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
10-methoxy-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(furan-3-ylmethyl)-N,6-dimethyl-2-(morpholin-4-yl)pyrimidin-4-amine
1-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]azetidin-3-yl}piperidine
1-[4-(4-hydroxy-4-phenylpiperidine-1-carbonyl)piperidin-1-yl]-2-methoxyethan-1-one
(3R,5S)-N-butyl-1-(2-methylpropyl)-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N-butyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(2-hydroxyphenyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
7-fluoro-4-[4-(1-methylpiperidin-4-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-dihydrophthalazin-1-one
1-[(5-methylpyrazin-2-yl)methyl]-3-(2,4,6-trimethylpyridin-3-yl)urea
2-[methyl(pyrazin-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-hexyl-8-(3-hydroxypropanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
6,7-difluoro-3-(3-hydroxypropyl)-3,4-dihydroquinazolin-4-one
N3-cyclohexyl-N5-cyclooctyl-N3-methyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-{[(2,6-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl][(5-methylthiophen-2-yl)methyl]amine
N-(1H-1,2,3-benzotriazol-5-yl)-4-[(propan-2-yl)sulfamoyl]benzamide
methyl 2-[1-(1H-imidazol-2-ylmethyl)-3-oxopiperazin-2-yl]acetate
2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]oxane-4-carboxamide
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-3-fluoro-N-(pyridin-3-ylmethyl)benzamide
3-(6-methoxypyridin-3-yl)-4-methylbenzoic acid
[(3R,4R)-1-(2-aminopyrimidin-4-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3S,4R)-1-acetyl-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
5-(4-chlorophenyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-1,2,4-triazin-3-amine
ethyl 4-(2-oxo-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-1-yl)piperidine-1-carboxylate
1-(1-methylpiperidin-4-yl)-N-(2-methylpropyl)piperidine-3-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(methylsulfanyl)ethan-1-one
4-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
5-{[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]methyl}thiophene-2-carboxylic acid