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(1S,5R)-3-[2-(methylamino)-1,3-thiazole-4-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(2-fluoro-5-methoxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(3-methoxypyrazin-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
1-methanesulfonyl-N-[(2-methoxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(piperidin-1-yl)acetamide
N-methyl-2-[4-({[1-(piperidin-1-ylmethyl)cyclohexyl]carbamoyl}amino)phenyl]acetamide
(3aS,6aS)-2-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,7aR)-1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
4-ethyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpyrimidine
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
[(4aS,8aR)-6-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N-(1-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}ethyl)-N-methylpropanamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(prop-2-en-1-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-cyclooctyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2-oxo-N-(oxolan-2-ylmethyl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-methylpropan-1-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}benzamide
6-cyclopropyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
ethyl 1-(1-{1,3-dioxo-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)piperidine-4-carboxylate
4-[2-(4-fluorophenyl)morpholin-4-yl]butan-1-ol
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(1,4-dioxan-2-ylmethyl)methylamine
1,3-dimethyl-2,6-dioxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(thiolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(dimethylamino)-2-[2-(1H-pyrrol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
N-[3-(1H-indazol-5-yl)phenyl]acetamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylthiophene-2-carboxamide
2-methyl-8-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-(4-chloro-2-methylphenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-(3,4,5-trifluorophenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-methyl-N-[3-(pyridin-3-yl)propyl]-1H-imidazole-2-carboxamide
4-methoxy-N-(2-methoxyethyl)-N-{[2-(2-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N,3-dimethyl-4-oxo-N-[3-(piperidin-1-yl)propyl]-3,4-dihydrophthalazine-1-carboxamide
N-(2H-1,3-benzodioxol-4-ylmethyl)-5-(1-benzyl-1H-pyrazol-3-yl)-4-methyl-1,3-thiazol-2-amine
1-(2-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)piperidin-2-one
2-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
dimethyl(2-{2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-({1-[(1-ethylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-3,3-dimethylpiperazin-2-one
4-[(2S)-1-[(5-butylthiophen-2-yl)methyl]pyrrolidine-2-carbonyl]morpholine
2-cyclopentyl-N-[(3-methyloxetan-3-yl)methyl]-2-phenylacetamide
2-(2-{[(1-cyclopropyl-1H-imidazol-5-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
1-[2-(pyrrolidin-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[6-amino-5-cyano-4-(3-hydroxyphenyl)pyridin-2-yl]benzoic acid
1-[2-(5-chloro-2-methoxypyridin-4-yl)pyrimidin-4-yl]pyrrolidin-3-ol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(piperidin-1-yl)acetamide
3-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
1-{4-[(1-benzothiophen-5-ylmethyl)amino]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one