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{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(cyclopropylmethyl)propylamine
1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)azepane
ethyl 2-[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]pyridine-3-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-4-(furan-2-carbonyl)piperazine-1-carboxamide
5,6-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
1-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2-{pyrazolo[1,5-a]pyridin-7-yl}-4-(trifluoromethyl)pyridine
N-[(3S,4R)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
6-(dimethylamino)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]acetamide
3-(azocan-1-yl)-N-[2-(ethylsulfanyl)ethyl]propanamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
1-(naphthalen-1-ylmethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
5-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-2-methoxybenzoic acid
4-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-2-methylquinoline
2-[4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]pyridine-3-carboxamide
4-[(2,4-dimethoxyphenyl)methyl]-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1-methyl-1H-imidazol-2-yl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine
5-(4-methylphenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-3-carboxamide
7-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-cyclopropyl-9-[(4-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-benzyl-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-(1,3-benzothiazol-2-ylmethyl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2-fluorophenyl)methyl]-3-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}propanamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylprop-2-en-1-yl)amine
2-methyl-5-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-ethyl-1H-pyrrole-2-carboxamide
3-[(5-chlorothiophen-2-yl)methyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
6-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[3-(2,6-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
2-[3,5-dimethyl-4-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-sulfonamido)-1H-pyrazol-1-yl]acetic acid
2-{2-[(2,3-dihydro-1H-inden-2-yl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
ethyl 3-({1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)propanoate
N-cyclopropyl-2-(dimethylamino)-2-(2-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]acetamide
N-(cyclopent-3-en-1-yl)-7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
N,N-diethyl-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopropyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
1-(4-chlorophenyl)-N-({1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(2-methyl-1,3-benzoxazole-6-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(4-fluorophenyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxopyrrolidin-1-yl)acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(3,3,3-trifluoropropanamido)acetic acid
N,N-diethyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2R,4S)-4-hydroxy-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-2-carboxylic acid
1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
3-{4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}-1,2-benzothiazole