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7-(5-propyl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-methyl-N-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}ethyl)propanamide
(3S)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-1-yl)ethyl]acetamide
1-cyclopentyl-4-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetyl}piperazin-2-one
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-[1-(furan-2-carbonyl)piperidin-4-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[2-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
3-[1-(3-hydroxypropanoyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-cyclopropyl-2-({1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
1-{3-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidine
N-(3,4-dimethoxyphenyl)-5-{4-hydroxy-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
2-methoxy-3-[5-(piperidine-1-carbonyl)pyridin-2-yl]quinoline
1-methyl-3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
4-[(5-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-propylpiperidine
N-(1-phenylpiperidin-4-yl)-3-(pyridin-4-yl)propanamide
6-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(propan-2-yl)pyrimidin-4-amine
butyl (1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
2-hydroxy-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,3-dimethylbutanamide
[5-chloro-7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[4-(difluoromethoxy)-2-methylphenyl]-2-(2-methoxyethyl)morpholine-4-carboxamide
4-(5-chlorothiophene-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
5-ethyl-N-methyl-N-[4-(morpholin-4-yl)butyl]pyrimidin-2-amine
(3S,4S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-methylpiperidine-3,4-diol
(2R,6S)-4-(6-chloro-3-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)-2,6-dimethylmorpholine
3-(2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,5-dimethoxyphenyl)pyridine-3-carbonitrile
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
5-methanesulfonyl-2-methyl-4-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]pyrimidine
(4aR,8aR)-7-[(3,5-difluorophenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
4-{4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazol-5-yl}phenol
N-cyclopentyl-1-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{5-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]thiophen-2-yl}ethan-1-one
2,4-dichloro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(quinolin-3-yl)oxan-4-yl]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3,5-dimethylbenzamide
(3S,9aR)-3-(4-aminobutyl)-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 1-(2-benzyl-1,3-benzoxazole-5-carbonyl)piperidine-2-carboxylate
2-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)-1,3-thiazole
1-(3-methylbenzenesulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-({[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1-phenylcyclopropanecarbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N1-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)piperidine-1,4-dicarboxamide
(3R,4S)-1-[1-(2-methoxyphenyl)piperidin-4-yl]-3,4-dimethylpiperidin-4-ol