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ethyl 4-(8-methyl-3-{[1-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)formamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
N-[(2S,4R,6R)-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-6-phenyloxan-4-yl]acetamide
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1H-pyrazole
N-(piperidin-4-yl)-1-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-(1H-pyrazol-3-yl)-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline
ethyl 1-(1H-indole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[2-(ethylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
8-{[5-(furan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{5-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepan-5-one
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[1-(2,5-dichlorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]butanoic acid
8-fluoro-2-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)quinolin-4-ol
1-{3-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]piperidin-1-yl}ethan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-oxopropanamide
2-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]amino}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-(quinolin-5-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2-methoxyethyl)-4-{[4-(methylamino)pyrimidin-2-yl]amino}pyrrolidin-2-one
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
(2-{[4-(1-methylazepane-2-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
3-methyl-5-{1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-2-yl}-1H-1,2,4-triazole
4-[6-(2-methyl-4-phenylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]morpholine
4-[1-(6-carbamoyl-2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]benzoic acid
5-benzyl-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1H-pyrazol-4-yl)ethyl]piperidin-2-one
2-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}pyridine
1-[4-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[3-(4-methoxyphenyl)-4-methyl-1H-pyrazol-1-yl]acetamide
(3S,4S)-4-methyl-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidine-3,4-diol
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-[({2-[cyclopentyl(methyl)amino]ethyl}(methyl)carbamoyl)amino]-3-methyl-N-(propan-2-yl)benzamide
N-benzyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]benzene-1-sulfonamide
N-ethyl-N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-cyclopropyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-ethoxyphenyl)methyl]acetamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-methoxy-3-methylphenyl)methyl]methylamine
7-methoxy-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzamide
3-(2-fluoro-3-methoxyphenyl)-4-methoxy-N-methylbenzamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperidin-4-ol
N-{[3-methyl-7-(4-phenylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}oxane-4-carboxamide
3-ethyl-4-{3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazin-2-one
(3R,4R)-4-(2-methoxyethyl)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-3-methylpiperidin-4-ol
(2S)-N-(2-chloro-4-fluoro-5-methylphenyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
N-[2-(4-fluorophenyl)ethyl]-2-(6-hydroxy-1,4-oxazepan-4-yl)acetamide
2-(4-chlorophenyl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-4-yl)propyl]pyrimidin-2-amine
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-N-ethylpyrimidin-2-amine