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1-[4-(4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
3-(4-chlorophenyl)-1-(4-hydroxypiperidin-1-yl)-3-phenylpropan-1-one
(3R,4S)-4-cyclopropyl-1-(4-ethyl-5-methylpyrimidin-2-yl)pyrrolidin-3-amine
(3S,4S)-1-(2,3-dimethylquinoxaline-6-carbonyl)-4-methylpiperidine-3,4-diol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
(3R,4S)-1-(5-phenyl-1,3,4-thiadiazol-2-yl)-4-propylpyrrolidin-3-amine
(3aR,6aS)-2-methyl-5-(2-oxo-4-phenylbutanoyl)-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-butyl-N-(furan-2-ylmethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
(3S,4R)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-methylpiperidine-3,4-diol
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(3-phenoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-(oxolan-2-ylmethyl)-2-(phenylformamido)-N-(pyridin-2-ylmethyl)acetamide
2-methyl-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]-1H-imidazole-4-carboxamide
(4aR,7aS)-1-[(2-methoxy-4-methylphenyl)methyl]-4-(3-methylbutyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-chloro-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-{4-[2-(3-fluorophenyl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
(3S,4R)-4-(3-methoxyphenyl)-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidine-3-carboxylic acid
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-2-(pyridin-4-yl)quinoline
N-(5-acetamido-2-fluorophenyl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
N-(butan-2-yl)-5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-phenyl-3-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]propan-2-ol
5-(2-methoxyphenoxymethyl)-N-(2-oxopiperidin-3-yl)-1H-pyrazole-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-4-(hydroxymethyl)pyridine-2-carboxamide
2-butyl-6-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
3-cyclopropaneamido-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-benzoxazol-2-amine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(ethylamino)pyrimidine-5-carboxamide
5-[(4aS,8aR)-decahydroisoquinolin-2-yl]-1-(naphthalen-2-ylmethyl)azepan-2-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[methyl(propan-2-yl)amino]ethan-1-one
2-ethyl-5-(4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine
3-{[2-(1H-imidazol-4-yl)ethyl]amino}-N-(1-phenylethyl)propanamide
methyl 1-[(3R,5S)-1-[(3-chlorophenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-({[(4-fluorophenyl)methyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
N-[(3-fluoro-4-methylphenyl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[2-(3-methoxyphenyl)-1-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
1-[1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
[2-(4-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}phenoxy)ethyl]dimethylamine
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
3-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}phenol
3-(2,3-dimethoxy-5-methylphenyl)pyrazolo[1,5-a]pyrimidine
3-(4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenyl)prop-2-yn-1-ol
N-[3-(cyclohexyloxy)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1,4-dithiepan-6-amine
N,N-dimethyl-2-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine