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(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine-2,4-diamine
5-{[2-(dimethylamino)ethyl]amino}-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[3-(1H-pyrazol-5-yl)phenyl]pyridine-3-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-phenoxybenzoyl)piperidine
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-ethyl-N-methyl-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-[2-(4-hydroxyphenyl)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
4-(3-butoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
(3aR,6aR)-2-cyclopropanecarbonyl-N-[2-(1H-imidazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}acetamide
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}sulfamoyl)-N-(pyridin-3-yl)benzamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-(propane-2-sulfonyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-({[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]amino}methyl)-5,8-dimethylquinolin-4-ol
4-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)but-3-yn-1-ol
4-(9-methoxy-7-oxo-3-{[4-(trifluoromethoxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)piperazin-2-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
1-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
1-(4-methoxyphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-[2-(methylsulfanyl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
(1R,5R)-3-(2,3-difluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-{2-[(4,6-dimethoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}-4-methyl-1,4-diazepane
1-(4-fluorophenyl)-4-[(4-methoxy-3-{2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
4-{[1-(2,3-dimethylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
1-{3-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
5-[(3-hydroxypyrrolidin-3-yl)methyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-({methyl[4-(morpholin-4-yl)butyl]amino}methyl)quinolin-4-ol
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
3-{[3-cyclopentyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(piperazin-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-[(4-hydroxyphenyl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)azetidine-2-carboxylic acid
(2E)-N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(4-methoxyphenyl)prop-2-enamide
2-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}morpholine
[(3-methoxyphenyl)methyl](methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
(2-methoxyethyl)[(4-methylphenyl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3,4-dimethoxyphenyl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]cyclopentane-1-carboxamide
N2-[(1S,3aS,6aS)-octahydropentalen-1-yl]-N4-methyl-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
7-(furan-3-ylmethyl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(2-chlorophenoxy)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]piperidin-2-one
2-(1-benzyl-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazin-2-yl)ethan-1-ol
1-methyl-4-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}-1,4-diazepane
5-methoxy-1-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide