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2-{[(4-fluorophenyl)methyl](methyl)amino}-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
3-{[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
N4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl]acetamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}pyridine-3-sulfonamide
3-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4-fluorophenyl)benzamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-(3-hydroxy-2-methylbenzoyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
(3S,7S)-5-(2-amino-6-methylpyrimidin-4-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-2-phenylethane-1,2-dione
methyl 1-[(3R,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(quinolin-6-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
ethyl 4-{3-[(1H-indazol-3-ylformamido)methyl]piperidin-1-yl}piperidine-1-carboxylate
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(3-cyanophenyl)methyl]-4-phenoxypiperidine-4-carboxylic acid
[2-(4-cyclohexanecarbonylmorpholin-2-yl)ethyl]dimethylamine
(1S,9aR)-1-({4-[3-(furan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-octahydro-1H-quinolizine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-5-propyl-1,2-oxazole-3-carboxamide
[(3-benzyl-1H-1,2,4-triazol-5-yl)(3-methylphenyl)methyl]dimethylamine
1-[(1R,5R)-6-{[4-(cyclopentyloxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-benzoyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)pyridine-2-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidine-3-carboxylic acid
2-[(propan-2-yl)amino]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}benzamide
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-methyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
1-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}cyclopropan-1-amine
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-{4-oxo-4-[4-(2-phenoxyethyl)piperazin-1-yl]butyl}piperidin-2-one
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
(1S,5R)-6-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-5-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(2S,4R)-4-amino-N-methyl-1-[2-(pyridin-4-yl)ethanesulfonyl]pyrrolidine-2-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
[2-(1H-imidazol-4-yl)ethyl]({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
N-methyl-N-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]methanesulfonamide
N-(2-{7-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
[4-({[4-(dimethylamino)-5-fluoropyrimidin-2-yl](methyl)amino}methyl)oxan-4-yl]methanol
N5-cyclooctyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(methylsulfanyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
[(2S,4R)-4-(dimethylamino)-1-[(6-phenoxypyridin-3-yl)methyl]pyrrolidin-2-yl]methanol
1-cyclopentyl-4-[4-(2-fluoro-4-methoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[4-(2-hydroxy-2-phenylpropanamido)phenyl]pentanamide
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2-methylphenyl)ethan-1-one
N,1-dimethyl-N-(1-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-3-carboxamide