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N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
1-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}piperidin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
1-butyl-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperazin-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-4-(3-phenylpropyl)piperazin-2-one
N-cyclopropyl-5-(quinoline-8-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-2-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
N-[(2,3-dimethoxyphenyl)methyl]-4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
(1s,4r)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-propylcyclohexane-1-carboxamide
3-methyl-7-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-(1-carbamoylcycloheptyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
3-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide
3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-1-(morpholin-4-yl)propan-1-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
6-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-amine
methyl 2-[4-(1-acetylpiperidin-4-yl)-3-methyl-2-oxopiperazin-1-yl]acetate
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalene-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-fluoro-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[3-(6-hydroxy-1,4-oxazepan-4-yl)-3-oxopropyl]-2,3-dihydro-1H-isoindol-1-one
2-[3-(propan-2-yloxy)phenyl]pyridine-4-carboxamide
(2E)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-(2,5-dimethoxybenzoyl)piperidine-4-carboxylate
1-[(2-fluorophenyl)methyl]-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]-1,4-diazepane
1-cyclohexanecarbonyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]morpholine
2-(methoxymethyl)-5-[(3-{2-[4-(1H-pyrazol-5-yl)phenyl]pyridin-4-yl}pyrrolidin-1-yl)methyl]pyrimidine
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
2-(3-fluorophenyl)-N-(4-{4-[(6-hydroxy-6-methylheptan-2-yl)amino]piperidin-1-yl}phenyl)acetamide
2-[methyl(quinolin-4-ylmethyl)amino]-2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]acetic acid
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxamide
4-{[4-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
6-(2-methoxyphenyl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyridazin-3-amine
1-[4-(3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(methylcarbamoyl)methyl]piperidin-4-yl}oxy)benzamide
1-{6-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]pyridin-3-yl}ethan-1-one
N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-amine
8-(1,3-benzothiazol-2-yl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane
1-{2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
[(1,2-dimethyl-1H-imidazol-5-yl)methyl]({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
1-methyl-3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
4-ethyl-3-{1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide