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(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
[3-(3-methylbut-2-en-1-yl)-1-(quinoxalin-2-yl)piperidin-3-yl]methanol
3-[4-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperazin-1-yl]propan-1-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[2-(2-fluorophenyl)ethyl]piperidine
N-[4-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
9-({4-[1-(dimethylamino)ethyl]phenyl}methyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-6-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-(3-hydroxy-3-phenylpropyl)-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
1-methyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
methyl 3-cyclobutaneamido-5-(cyclohexylamino)-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
4-(1-methyl-3-{4-[(thiophen-2-ylmethoxy)methyl]phenyl}-1H-1,2,4-triazol-5-yl)morpholine
2-(3-fluoro-2,4-dimethylphenyl)-1-[2-(2-methylpropanesulfonyl)ethyl]-1H-imidazole
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-[4-(trifluoromethoxy)phenyl]urea
(2R)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}oxolane-2-carboxamide
1-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
4-{5-[(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-(2-methoxyethyl)-9-[(2-methylnaphthalen-1-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-difluorophenyl)-1-(thiophen-3-ylmethyl)piperidin-3-amine
2-(2,4,6-trimethylphenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(3-acetamidophenyl)-3-(4-methyl-1,4-diazepan-1-yl)propanamide
4-benzyl-1-[(3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-oxazol-5-yl)methyl]piperidine
N-(2-{[(3R,5R)-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
2-[(2,6-dichlorophenyl)methyl]-5-(pyrrolidine-1-carbonyl)pyrimidin-4-ol
4-(1H-pyrrole-2-carbonyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazine-1-carboxamide
4-[({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
N-[(2,4-dichlorophenyl)methyl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(1-ethyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-2-one
4-ethyl-3-{[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-acetamido-4-fluorophenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
2-(4-fluorophenyl)-4-(2-propoxybenzoyl)morpholine
8-(3-hydroxypyridine-2-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
8-{[2-(5-methylfuran-2-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N,N-dimethylbenzamide
4-[1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-4-yl]thiomorpholine
(1R,5S,8S)-8-methoxy-N-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
1-(3-fluoropyridine-4-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(pyridin-3-yloxy)propyl]acetamide
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
4-methyl-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}pentan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,3-dicyclopropyl-1H-pyrazole-5-carboxamide
6-{4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-methoxy-3-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyrazine
1-(1,2-oxazole-3-carbonyl)-3-(thiophene-2-carbonyl)piperidine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2,5-dimethoxybenzene-1-sulfonamide