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1-cyclopentyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-5-oxopyrrolidine-3-carboxamide
1-{3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}-4-phenylpiperidine
2-methyl-3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
8-fluoro-2-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)quinoline
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-[1-(2-phenylethyl)-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-6-methoxypyrimidin-4-amine
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(4aS,8aR)-1-(carboxymethyl)-6-(2-phenylethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-methyl-6-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}pyrimidin-2-amine
(3S,4R)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
4-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperazine-2-carboxylic acid
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methylphenol
3-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
3-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[2-fluoro-3-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
3-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]benzoic acid
1-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(propan-2-yl)urea
methyl (2S,4R)-4-(dimethylamino)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
3-(2-hydroxyphenyl)-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-{2-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)-8-azabicyclo[3.2.1]octane-8-carboxamide
(2E)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-[(2S)-1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-4-methyl-1-oxopentan-2-yl]acetamide
5-(8-methoxyquinolin-5-yl)pyridin-3-amine
3-(2-methylphenyl)-3-phenyl-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
1-(6-fluoropyridin-3-yl)-3-methyl-3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]urea
2-methoxyethyl 3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
8-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-{2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-(2-ethoxyethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-[1-(7-chloroquinoxalin-2-yl)piperidin-3-yl]ethan-1-amine
2-(4-fluorophenoxymethyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
(3S,9aR)-3-benzyl-8-(4-chlorobenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
6-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(benzyloxy)benzoyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(dimethylamino)-2-(3-fluorophenyl)ethan-1-one
3-{[2-(1-benzyl-3-oxopiperazin-2-yl)acetamido]methyl}-N-methylbenzamide
4-[(5-methylfuran-2-yl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
N-{[1-(1,4-dithiepan-6-yl)pyrrolidin-3-yl]methyl}methanesulfonamide