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3-{5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(2-hydroxyethyl)propanamide
3-(1-methylpiperidin-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}propanamide
3-methyl-7-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(6-aminopyridin-3-yl)-2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]acetic acid
2-(3-methylphenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-[methyl({4-methyl-5-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-(2-chloro-4-fluorobenzoyl)-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
(2S,4R)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(pyrrolidine-1-carbonyl)piperidine
2,3,6-trimethyl-N-(2-oxopyrrolidin-3-yl)quinoline-4-carboxamide
4-hydroxy-2-methyl-N-[2-(2-oxopyrrolidin-1-yl)ethyl]benzamide
N-(2,3-dihydro-1H-inden-2-yl)-N,5,7-trimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-aminoethyl)-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-4-phenyl-1-(1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
2,4,5-trimethoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
4-(2,4-dioxoimidazolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
2-{4-[4-(dimethylcarbamoyl)phenyl]phenyl}acetic acid
2-(1-cyclopentyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl)ethan-1-ol
3-(3-methoxypropyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxylic acid
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-6-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-methyl-N-{1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-indazole-3-carboxamide
2-(4-chlorophenyl)-4-(6-cyclopropylpyrimidin-4-yl)morpholine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(3-cyclopentylpropyl)methylamine
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}prop-2-enamide
2-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-cyclohexyl-2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{3-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]morpholin-4-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
2-(2-methoxy-4-methylphenoxymethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazole
N-(1,3-benzoxazol-2-ylmethyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[1-(3-methylbut-2-en-1-yl)-4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-cyclopropyl-6-(2-fluorophenyl)-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-[(2,3-dimethoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrimidin-2-amine
(3S,4S)-4-cyclopropyl-1-(3,4-difluorobenzoyl)pyrrolidine-3-carboxylic acid
N-[2-(pyridin-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
1-[(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)methyl]-1H-pyrazole
N-[2-(ethanesulfonyl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[(2-chlorophenyl)methyl]-6-methyl-4-oxo-N-(propan-2-yl)-1,4-dihydroquinoline-3-carboxamide
N-methyl-2-[(3R,4S)-3-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamido]-4-propylpyrrolidin-1-yl]acetamide