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6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-N-[(1-hydroxycyclohexyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amine
5-chloro-N-{2-[(2-ethylphenyl)carbamoyl]phenyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{1-[1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[2-(pyridin-4-yl)ethyl]benzamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-3-phenoxypropan-1-one
3-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
N-(5-methyl-1,2-oxazol-3-yl)-3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazole-5-carboxamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-methyl-2-(morpholin-4-yl)propan-1-one
1-(3-cyano-4-ethoxyphenyl)-3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
2-methoxy-N-{1-methyl-7-[3-(3-methylbutanoyl)piperidine-1-carbonyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl}acetamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(2,3,6-trifluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]pyrazine
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
6-(3-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-N-(pyrimidin-4-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-amino-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(dimethylamino)-2,2-dimethylpropyl]acetamide
1,2-dimethyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
1-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-phenylethane-1,2-dione
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]acetamide
3-[(4-cyanopiperidin-1-yl)sulfonyl]-N-(oxolan-3-ylmethyl)benzamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclohexyl-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N5-[2-(cyclohex-1-en-1-yl)ethyl]-N3-(2-hydroxyethyl)-1-[(2-methoxyphenyl)methyl]-4-oxo-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(4-fluorophenyl)-3-(pyrrolidin-1-yl)-1,2,4-triazine
7-fluoro-3-methyl-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-indole-2-carboxamide
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}azetidin-3-yl)-2-methylpiperidine
3-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-4-carboxylic acid
4-(cyclohexylmethyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,4-diazepan-5-one
3-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2-dimethyl-1H-indole
N-{1-[3-(carbamoylmethyl)-1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]butyl}acetamide
1-methyl-4-[3-(methylsulfanyl)propyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)oxane-4-carboxamide
1-({4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-5-methyl-1H-1,2,3,4-tetrazole
1-[6-(dimethylcarbamoyl)pyrazin-2-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(2-phenylethyl)-7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[3-(2-cyclohexylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrazine
1-[(4-{[1-(furan-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-phenylpiperidine
5-ethyl-4-[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]pyrimidin-2-amine
2-[3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(3R,4S)-4-cyclopropyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)pyrrolidin-3-amine
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(pyridin-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-propyl-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrimidine
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-5-carboxamide
N-{[(2S,4S)-1-[(2R)-2-amino-3-(1H-indol-3-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide