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7-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2S,4R)-4-amino-N,N-diethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-[(3-fluorophenyl)methyl]-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
7-chloro-N-(2-hydroxyethyl)-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-indole-2-carboxamide
4-[(1R,7S)-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine-4-carboxamide
5-methoxy-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
(1S,2S,9R)-11-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)cyclobutanamine
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-5-carboxamide
4-[1-(3-chloro-4-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
4-[(2-chlorophenyl)methyl]-1-[(2E)-2-methylbut-2-enoyl]-1,4-diazepan-5-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1-cyclobutanecarbonyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
N-methyl-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]pentanamide
N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[(3-methoxyphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}morpholine
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2-chlorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(4aR,8aS)-1-[3-(dimethylamino)propyl]-6-(furan-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[2-(4-methoxyphenyl)ethyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
4-(1-acetylpiperidin-4-yl)-3-butyl-1-methylpiperazin-2-one
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-benzyl-N-methylpiperidin-3-amine
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(3-phenylpropyl)morpholine
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[3-(1H-pyrazol-1-yl)propyl]-1,4-diazepan-5-one
4-(quinolin-3-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-1-{4-[2-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-1-ol
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-4-propyl-1,2,3-thiadiazole
N-methyl-N-(2-methylpropyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
2-[3-({4-[5-(3-fluorophenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-[(2-fluorophenyl)methyl]-1-[3-(1H-indol-3-yl)propanoyl]-1,4-diazepan-5-one
3-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(4-chlorophenyl)-2-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-phenyl-8-(quinolin-4-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-{[4-(1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N-methylpyridin-2-amine
N-(9H-fluoren-9-yl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N,N-dimethyl-3-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)propanamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(2R,6R)-4-(1,3-dihydroxypropan-2-yl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(1-{[3-(2-aminoethyl)phenyl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-(thiophen-2-yl)-1,2,4-oxadiazole
4-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]piperazine-2-carboxylic acid
1-[(3-methoxyphenyl)methyl]-4-{3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanoyl}piperazin-2-one