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2-{3-oxo-9-[(1-propyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-(2-fluorophenyl)-3-(2-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
1-(3-acetylphenyl)-3-(2,2-dimethyloxan-4-yl)-3-ethylurea
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
3-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
2-(2-fluorophenoxymethyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,3-oxazole-4-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
[(2S)-1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl]methanol
8-[(2-fluoro-4-methoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-fluorophenyl)-3-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
1-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]isoquinoline
5-cyclopropyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-1-[(4Z)-hept-4-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-({2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-N,N-dimethylbenzamide
2-methyl-6-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}pyridine
(3R,4R)-4-(azepan-1-yl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
(5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-butyl-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
5-({[5-(2,5-dimethylfuran-3-yl)-1,2,4-triazin-3-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1,3-diazinane-2,4-dione
(4aR,8aR)-2-methanesulfonyl-7-[(3-methylquinoxalin-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
7-chloro-3-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
3-({3-cyclopropyl-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methoxy)-2-ethyl-6-methylpyridine
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
2-(morpholin-4-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(pyridin-3-yl)acetamide
2-[4-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-3-(propan-2-yl)piperazin-2-one
2-(5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-2-one
(2E)-1-[3-(4-chlorobenzoyl)piperidin-1-yl]-4-methylpent-2-en-1-one
4-chloro-2-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenol
N-(furan-3-ylmethyl)-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-methyl-3-{4-[1-(piperidin-1-yl)ethyl]phenyl}benzoic acid
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
4-{1-[1-(5-propylthiophene-3-carbonyl)piperidin-4-yl]ethyl}morpholine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-fluorophenyl)ethan-1-one
N-(1-methoxybutan-2-yl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
2-amino-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
6-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
3-(5-{2-[4-(propan-2-yl)phenyl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-N-methyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-amine
methyl 3-cyclohexyl-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
N-(4-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one