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N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
2,5,7-trimethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]quinoline-4-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-(1-benzoylpiperidin-4-yl)-N-(2-methoxyethyl)piperidine-3-carboxamide
N4-[1-(3,4-dimethylphenyl)ethyl]-5-ethylpyrimidine-2,4-diamine
4-[(dimethylamino)methyl]-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)azepan-4-ol
4-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-(2-hydroxypropan-2-yl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
ethyl 2-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
4-methyl-2-{2-[3-(morpholin-4-yl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
(butan-2-yl)(pyridin-3-ylmethyl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
1-(3-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
3-amino-N-(butan-2-yl)-N-cyclopentylpropanamide
(1S,5R)-3-[2-(4-fluorophenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aS)-2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-decahydroisoquinolin-4a-ol
6-(2-chlorophenyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
(3S,4R)-1-[methyl(propan-2-yl)sulfamoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-1-(2-methylpropyl)-5-{[3-(pyridin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[3-(2,2-dimethylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
N-(3-ethoxypyridin-2-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}benzamide
1-(4-chloro-3-fluorobenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
2-[(1S,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
[1-(3-{[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}propyl)piperidin-2-yl]methanol
N-(2-fluoro-4-methylphenyl)-2-{[1-(piperidin-1-yl)propan-2-yl]amino}acetamide
N-{[1-(pyridazine-4-carbonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
2-(dimethylamino)-8-{3-[(dimethylamino)methyl]-4-methoxyphenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-hydroxy-2-(3-methylphenyl)-N-[(3S)-2-oxoazepan-3-yl]pyrimidine-5-carboxamide
2-(3,4-dimethylphenoxy)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
1'-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
methyl 3-cyclobutaneamido-5-{[(2-methoxyphenyl)formamido]methyl}benzoate
1-(2,4-difluorophenyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-cyclopentyl-N-(3-methylbutyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-(4-fluorophenyl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}cyclopropane-1-carboxamide
1-(3-phenylpropyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-2-amine
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
5-cyclobutanecarbonyl-1'-[(2R)-pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(but-2-yn-1-yl)({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(furan-2-ylmethyl)amine
6-tert-butyl-2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2,3-dihydropyrimidine-4-carboxamide
1-[5-(1-carboxy-1-methylethyl)-4-(morpholin-4-yl)pyrimidin-2-yl]piperidine-4-carboxylic acid
(cyclohex-3-en-1-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(2S,4R)-4-amino-1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-N-ethylpyrrolidine-2-carboxamide
2-{[(3-methylpyridin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{4-[3-(4-chlorobenzoyl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N-[(1R,3R)-3-aminocyclopentyl]-4-pentylbenzene-1-sulfonamide
methyl 4-[4-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate