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methyl (2S,4R)-4-[3-(4-methylphenyl)propanamido]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxylate
N,N-diethyl-1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
(1-benzofuran-2-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
(3R,4S)-1-(2,3-difluoro-4-methylbenzoyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
methyl 3-{[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}propanoate
3-chloro-6-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]pyridine-2-carboxylic acid
{[(3S,4R)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
3-(oxolan-2-yl)-7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
6-(2-methylphenyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{5-[(4-hydroxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-ol
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidine
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(pyridin-3-yl)pyrimidine
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(2-methoxyethyl)-N-methyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
4-[4-(5-chlorothiophen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
methyl 3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
3-hydroxy-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
2-amino-3-ethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
{9-[3-(1H-pyrazol-1-yl)propyl]-3-(1H-pyrrole-2-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1'-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-methyl-4-{3-[3-(phenoxymethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
4-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}quinoline
N,N-dimethyl-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
6-[2-(naphthalen-1-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(2-fluoroethyl)-1H-imidazol-2-yl]-2-(naphthalen-1-yl)pyrimidine
N-{1-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
5-({2-[3-(3-carboxyphenyl)piperidin-1-yl]acetamido}methyl)furan-2-carboxylic acid
1-[(3-methylpyridin-2-yl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
methyl 3-cyclohexaneamido-6-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
2-ethyl-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-cyclopentyl-4-(1H-indol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-(diethylamino)-3-[2-methoxy-4-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(3ar,6ar)-N-[(1-benzylpiperidin-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
8-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-N-(thiophen-2-yl)piperidine-1-carboxamide
1,2-dimethyl-4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazine
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-4-(piperidin-1-yl)butan-1-one
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
6-methoxy-3-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1-benzofuran-2-carboxamide
N-[4-(4-{[3-(1H-imidazol-1-yl)-1-phenylpropyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
ethyl 5-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-(7-chloroquinolin-4-yl)-1H-pyrazole-4-carboxylate
N-[4-ethoxy-3-(trifluoromethyl)phenyl]-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
methyl 5-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)piperidin-3-amine
2-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}-2-(thiomorpholin-4-yl)acetic acid
2-{2-[(2-ethylbutyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid