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[(2S)-1-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)amine
2-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,2,3,4-tetrahydroisoquinoline
3-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
1-[(3,5-dimethylphenyl)methyl]-4-(4,6-dimethylpyridine-3-carbonyl)piperazin-2-one
N-[(4-hydroxyazepan-4-yl)methyl]-2-methyl-1,3-benzothiazole-6-carboxamide
8-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-cyclopentyl-N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1,4-diazepane-1-carboxamide
N-phenyl-4-{1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-amido}piperidine-1-carboxamide
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[({5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)sulfanyl]-4H-1,2,4-triazole
N-methyl-7-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
2-methoxy-4-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
1-(2-chloro-3-methylbenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
(3aS,6aS)-2-benzyl-5-[2-(4-methylpiperidin-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-[(4-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-fluorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-{[(3,4-difluorophenyl)carbamoyl]methyl}-2-(4-propanoylphenoxy)acetamide
2-{1-[(4-ethoxyphenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
4-methoxy-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
1-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)urea
2-[(3-propylmorpholin-4-yl)methyl]quinoline
1-[2-hydroxy-3-(2-methoxy-4-{[methyl(propyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
2-(1,2-benzoxazol-3-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}acetamide
N-{1-[7-(3-methylbut-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
3-{[4-(3-methoxypropyl)piperazin-1-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-ethyl-3-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}pent-4-enamide
ethyl 5-({[3-(2-phenylethyl)-1,2-oxazol-5-yl]formamido}methyl)furan-2-carboxylate
1-{[3-(3-phenoxyazetidine-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
2-(5-acetylthiophen-3-yl)-N-[3-(cyclohexylsulfanyl)propyl]acetamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)butan-1-one
3-ethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-pyrazole-5-carboxamide
6-chloro-4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
(1S,6R)-9-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2R,3R)-2-hydroxy-1'-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
4-{4-[(3-hydroxypropyl)(methyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
1-(4-{[3-(5-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}furan-2-yl)-1H-pyrazol-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(3-methoxyphenoxy)propan-1-one
2-[4-(1-benzofuran-2-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
2-(4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidin-1-yl)pyrimidine
N'1-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]cyclopropane-1,1-dicarboxamide
methyl 4-[(3-{[2-(3-fluorophenyl)acetamido]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]benzoate
3-methyl-4-oxo-N-(thiolan-3-yl)-3,4-dihydrophthalazine-1-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}morpholine
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-5-methyl-6-phenylpyridine-3-carbonitrile
4-amino-N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]pyridine-2-carboxamide